SCHEMBL24914244

SCHEMBL24914244

CCOCCN1CCC(F)(F)C1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.35
SLC6A4 P31645 1/20 0.35
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
OPRM1 P35372 2/20 0.32
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP14 P50281 1/20 0.32
S1PR4 O95977 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
S1PR5 Q9H228 1/20 0.31
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30
MCHR1 Q99705 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25497517 0.81 HRH3 (0.48) HRH3SLC6A4CYP2D6CYP2C19OPRM1
SCHEMBL12712697 0.81 CNR2 (0.37) HRH3SLC6A4MMP1MMP9MMP14
SCHEMBL6118897 0.80 HTR1A (0.37) HRH3SLC6A4CYP2D6OPRM1
SCHEMBL23841765 0.79 CYP2D6 (0.36) HRH3SLC6A4CYP2D6CYP2C19OPRM1
SCHEMBL9946182 0.79 S1PR1 (0.47) OPRM1S1PR4S1PR1S1PR3S1PR5
SCHEMBL6890281 0.78 S1PR4 (0.35) HRH3SLC6A4CYP2D6OPRM1S1PR4
SCHEMBL12872465 0.78 HRH3 (0.33) HRH3SLC6A4MCHR1
SCHEMBL14116874 0.78 HRH3 (0.42) HRH3SLC6A4OPRM1S1PR4S1PR1
SCHEMBL23158170 0.77 HRH3 (0.33) HRH3SLC6A4
SCHEMBL20331193 0.77 S1PR1 (0.50) S1PR4S1PR1S1PR3S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230019236-A1 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF CALICO LIFE SCIENCES LLC (US) 2023-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230019236-A1 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF PTPN1, PTPN2, PTPN18 HRH3 4595/4885SLC6A4 3966/4885CYP2D6 3885/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.