SCHEMBL24918232

SCHEMBL24918232

C[C@@H]1C(=O)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
NR1H2 P55055 1/20 0.38
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
MAPK1 P28482 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
HPGD P15428 1/20 0.36
ATM Q13315 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2395205 1.00 USP2 (0.39) USP2SMN1; SMN2HSD17B10KDM4EMAPT
SCHEMBL16224559 1.00 USP2 (0.39) USP2SMN1; SMN2HSD17B10KDM4EMAPT
SCHEMBL3805159 0.90 HSD17B10 (0.42) HSD17B10CHRM2CHRM1CHRM3HPGD
SCHEMBL4766170 0.90 HSD17B10 (0.42) HSD17B10CHRM2CHRM1CHRM3HPGD
SCHEMBL22120434 0.89 HSD17B10 (0.41) HSD17B10HPGD
SCHEMBL22128107 0.89 HSD17B10 (0.41) HSD17B10HPGD
SCHEMBL31066400 0.82 MAPK1 (0.39) USP2SMN1; SMN2HSD17B10KDM4EMAPT
SCHEMBL15797129 0.82 MAPK1 (0.39) USP2SMN1; SMN2HSD17B10KDM4EMAPT
SCHEMBL30867786 0.82 MAPK1 (0.39) USP2SMN1; SMN2HSD17B10KDM4EMAPT
SCHEMBL22820950 0.81 NPC1 (0.38) USP2SMN1; SMN2HSD17B10NR1H2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260125386-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF KRAS THERAS INC (US) 2026-05-07 US disclosed
US-12606572-B2 Substituted heterocycles and uses thereof KUMQUAT BIOSCIENCES INC. (US) 2026-04-21 US disclosed
EP-4724445-A1 SUBSTITUTED HETEROCYCLES AND USES THEREOF Kumquat Biosciences Inc. (US) 2026-04-15 EP disclosed
US-20260042764-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF KRAS THERAS INC (US) 2026-02-12 US disclosed
US-20260028357-A1 SUBSTITUTED HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC (US) 2026-01-29 US disclosed
US-12528818-B2 Compositions and methods for inhibition of RAS LEIDOS BIOMEDICAL RESEARCH, INC. (US) 2026-01-20 US disclosed
WO-2025264645-A1 SODIUM CHANNEL BLOCKING COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE LATIGO BIOTHERAPEUTICS, INC. (US) 2025-12-26 WO disclosed
US-20250270225-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS NNSA 2025-08-28 US disclosed
EP-4565579-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF KRAS Theras, Inc. (US) 2025-06-11 EP disclosed
WO-2024254334-A1 SUBSTITUTED HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC. (US) 2024-12-12 WO disclosed
US-20240300964-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS THERAS, INC. 2024-09-12 US disclosed
EP-4373822-A2 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS Theras Inc. (US) 2024-05-29 EP disclosed
CN-117916238-A Compositions and methods for inhibiting RAS 瑟拉斯有限公司 2024-04-19 CN disclosed
WO-2023004102-A2 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS THERAS, INC. (US) 2023-01-26 WO disclosed
WO-2023004102-A2 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS THERAS, INC. (US) 2023-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12606572-B2 Substituted heterocycles and uses thereof KRAS, HRAS, MYC USP2 3471/4885SMN1; SMN2 1611/4885HSD17B10 2162/4885
US-20250270225-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS KRAS, NRAS, HRAS USP2 673/4885SMN1; SMN2 2490/4885HSD17B10 2767/4885
US-20260125386-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF KRAS KRAS, NRAS, HRAS USP2 1517/4885SMN1; SMN2 1405/4885HSD17B10 3903/4885
US-20240300964-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS KRAS, NRAS, HRAS USP2 673/4885SMN1; SMN2 2490/4885HSD17B10 2767/4885
US-20260042764-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF KRAS KRAS, NRAS, HRAS USP2 2112/4885SMN1; SMN2 2830/4885HSD17B10 1872/4885
US-12528818-B2 Compositions and methods for inhibition of RAS KRAS, NRAS, HRAS USP2 1068/4885SMN1; SMN2 654/4885HSD17B10 2660/4885
US-20260028357-A1 SUBSTITUTED HETEROCYCLES AND USES THEREOF KRAS, HRAS, MYC USP2 3471/4885SMN1; SMN2 1611/4885HSD17B10 2162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.