SCHEMBL2491914

SCHEMBL2491914

CCC1[C@H](N(C)c2nc(-c3ccncc3)cc(=O)n2C)CCCN1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.41
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2491257 0.89 GSK3B (0.47) GSK3BCYP2D6
SCHEMBL2488119 0.81 GSK3B (0.44) GSK3BCYP1A2CYP2D6
SCHEMBL2490282 0.81 GSK3B (0.44) GSK3BCYP1A2CYP2D6
SCHEMBL3749271 0.77 GSK3B (0.43) GSK3BCYP1A2CYP2D6
SCHEMBL2491912 0.74 GSK3B (0.40) GSK3B
SCHEMBL2488072 0.74 GSK3B (0.45) GSK3BCYP1A2CYP2D6
SCHEMBL2489224 0.74 GSK3B (0.45) GSK3BCYP1A2CYP2D6
SCHEMBL2403922 0.74 GSK3B (0.54) GSK3BCYP1A2CYP2D6
SCHEMBL2527052 0.74 MAP4K4 (0.41) GSK3BCYP1A2CYP2D6
SCHEMBL2490162 0.74 GSK3B (0.47) GSK3BCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2057141-B1 PYRIMIDONE COMPOUNDS AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2011-10-26 EP disclosed