SCHEMBL24920532

SCHEMBL24920532

COCc1cnc(N2CCOCC2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.44
ALDH1A1 P00352 7/20 0.44
LMNA P02545 2/20 0.44
HTT P42858 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HSD17B10 Q99714 3/20 0.42
HPGD P15428 3/20 0.42
KDM4E B2RXH2 3/20 0.42
MAPT P10636 2/20 0.42
GAA P10253 2/20 0.42
MEN1 O00255 1/20 0.42
RECQL P46063 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CNR2 P34972 3/20 0.41
MTOR P42345 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP11B1 P15538 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9925951 0.83 ALDH1A1 (0.46) CYP2C19ALDH1A1LMNAHTTHSD17B10
SCHEMBL30922273 0.79 CNR2 (0.47) CYP2C19ALDH1A1LMNAHTTHSD17B10
SCHEMBL24921793 0.78 ALDH1A1 (0.46) CYP2C19ALDH1A1LMNAHTTL3MBTL1
SCHEMBL18885167 0.77 CYP11B1 (0.56) CYP2C19ALDH1A1LMNAHTTL3MBTL1
SCHEMBL10333903 0.77 CYP2C19 (0.61) CYP2C19ALDH1A1LMNAHTTL3MBTL1
SCHEMBL24921465 0.76 CYP2C19 (0.59) CYP2C19ALDH1A1LMNAHTTHSD17B10
SCHEMBL807298 0.74 ALDH1A1 (0.54) CYP2C19ALDH1A1LMNAHTTHSD17B10
SCHEMBL19534370 0.74 MTOR (0.39) ALDH1A1LMNAHTTL3MBTL1HSD17B10
SCHEMBL24921115 0.74 PIK3CD (0.44) CYP2C19ALDH1A1LMNAHTTHSD17B10
SCHEMBL1271706 0.73 ALDH1A1 (0.56) CYP2C19ALDH1A1LMNAHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed