SCHEMBL2492729

SCHEMBL2492729

CCOc1ccc(C)nc1C(=O)N1CCCCC1Cc1nc2c(C)cccn2c1Cl

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 12/20 0.43
HCRTR1 O43613 10/20 0.43
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
REN P00797 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2487836 1.00 HCRTR2 (0.43) HCRTR2HCRTR1ALDH1A1MAPK1MEN1
Hydrochloric Acid SCHEMBL2532203 0.99 HCRTR2 (0.43) HCRTR2HCRTR1ALDH1A1MAPK1MEN1
SCHEMBL2489774 0.93 HCRTR1 (0.43) HCRTR2HCRTR1ALDH1A1MAPK1REN
SCHEMBL2489769 0.93 HCRTR1 (0.43) HCRTR2HCRTR1ALDH1A1MAPK1REN
Hydrochloric Acid SCHEMBL2512752 0.92 HCRTR1 (0.42) HCRTR2HCRTR1ALDH1A1MAPK1REN
SCHEMBL2488664 0.85 HCRTR1 (0.44) HCRTR2HCRTR1ALDH1A1MAPK1MEN1
SCHEMBL2488670 0.85 HCRTR1 (0.44) HCRTR2HCRTR1ALDH1A1MAPK1MEN1
Hydrochloric Acid SCHEMBL2512388 0.84 HCRTR1 (0.43) HCRTR2HCRTR1ALDH1A1MAPK1MEN1
SCHEMBL4167405 0.81 ALDH1A1 (0.38) ALDH1A1MAPK1MEN1KMT2A
SCHEMBL2124396 0.78 PDE8B (0.41) HCRTR2ALDH1A1MEN1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379550-A1 PIPERIDINE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS Glaxo Group Limited (GB) 2011-10-26 EP disclosed
WO-2010072722-A1 PIPERIDINE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS GLAXO GROUP LIMITED (GB) 2010-07-01 WO disclosed