SCHEMBL24928529

SCHEMBL24928529

CC1CCC(Br)SC(N)=N1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.42
NOS2 P35228 5/20 0.42
NOS3 P29474 4/20 0.42
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
KMT2A Q03164 1/20 0.36
THRB P10828 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
GABRA5 P31644 2/20 0.31
GABRB2 P47870 2/20 0.31
GABRR1 P24046 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3191452 0.67
SCHEMBL13479874 0.67
Hydrochloric Acid SCHEMBL3178761 0.65 NOS1 (0.46) NOS1NOS2NOS3MEN1CYP1A2
Hydrochloric Acid SCHEMBL1922632 0.65
SCHEMBL9060276 0.64
Bromide SCHEMBL9060815 0.62 NOS1 (0.47) NOS1NOS2NOS3MEN1CYP1A2
SCHEMBL6330626 0.61
SCHEMBL8401014 0.59
Hydrochloric Acid SCHEMBL19667261 0.58
SCHEMBL8299940 0.58 NOS1 (0.64) NOS1NOS2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023009982-A1 SMALL MOLECULE INHIBITION OF DEUBIQUITINATING ENZYME JOSEPHIN DOMAIN CONTAINING 1 (JOSD1) AS A TARGETED THERAPY FOR LEUKEMIAS WITH MUTANT JANUS KINASE 2 (JAK2) DANA-FARBER CANCER INSTITUTE, INC. (US) 2023-02-02 WO disclosed