SCHEMBL24933856

SCHEMBL24933856

CC(C)Oc1ccncc1COc1ccc(-c2cc(C(N)=O)c(=O)[nH]c2C(F)(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 5/20 0.39
MKNK2 Q9HBH9 5/20 0.39
HSD17B1 P14061 3/20 0.37
HSD17B2 P37059 3/20 0.37
CSF1R P07333 2/20 0.35
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
IRAK4 Q9NWZ3 6/20 0.34
CDC7 O00311 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30240731 0.91 PARP10 (0.41) MKNK1MKNK2HSD17B1HSD17B2CDK5
SCHEMBL24933028 0.91 PARP10 (0.41) MKNK1MKNK2HSD17B1HSD17B2CDK5
SCHEMBL30240778 0.90 MKNK1 (0.43) MKNK1MKNK2HSD17B1HSD17B2CSF1R
SCHEMBL24933882 0.90 MKNK1 (0.43) MKNK1MKNK2HSD17B1HSD17B2CSF1R
SCHEMBL24933735 0.87 HSD17B1 (0.41) MKNK1MKNK2HSD17B1HSD17B2CDK5
SCHEMBL30240751 0.87 HSD17B1 (0.41) MKNK1MKNK2HSD17B1HSD17B2CDK5
SCHEMBL24933386 0.84 CDC7 (0.38) MKNK1MKNK2HSD17B1HSD17B2CDK5
SCHEMBL24933607 0.82 HSD17B2 (0.39) HSD17B1HSD17B2CDK5CDK5R1
SCHEMBL24933406 0.82 HSD17B1 (0.41) HSD17B1HSD17B2CDK5CDK5R1
SCHEMBL30240675 0.82 HSD17B1 (0.41) HSD17B1HSD17B2CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP claimed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN claimed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO claimed
EP-4373809-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS Novartis AG (CH) 2024-05-29 EP disclosed
CN-117980292-A Substituted pyridone compounds for the treatment of orthomyxoviral infections 诺华股份有限公司 2024-05-03 CN disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed
WO-2023002443-A1 SUBSTITUTED PYRIDONE COMPOUNDS USEFUL TO TREAT ORTHOMYXOVIRUS INFECTIONS NOVARTIS AG (CH) 2023-01-26 WO disclosed