SCHEMBL24947181

SCHEMBL24947181

COC(=O)c1ccc(C(F)(F)F)c2cc(C)oc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 6/20 0.43
NOTUM Q6P988 3/20 0.43
CYP1A1 P04798 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP1B1 Q16678 1/20 0.41
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 1/20 0.36
CES2 O00748 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK4 Q16654 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
KDM4E B2RXH2 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12566233 0.78 ALDH1A1 (0.40) ALDH1A1HPGDHSD17B10CA12CA1
SCHEMBL24947159 0.78 ABL1 (0.43) ALDH1A1HPGDHSD17B10CA12CA1
SCHEMBL29967405 0.77 CFTR (0.44) CFTRNOTUMALDH1A1HPGDHSD17B10
SCHEMBL28878138 0.77 CFTR (0.44) CFTRNOTUMALDH1A1HPGDHSD17B10
SCHEMBL2635958 0.75 CYP1A1 (0.43) NOTUMCYP1A1CYP1A2CYP1B1ALDH1A1
SCHEMBL28731299 0.75 GAA (0.44) CYP1A2ALDH1A1HPGDCA12CA1
SCHEMBL27706769 0.73 BRD4 (0.47) CFTRNOTUMALDH1A1HPGDHSD17B10
SCHEMBL12566234 0.73 GSK3B (0.47) CYP1A2ALDH1A1HPGDHSD17B10CA12
SCHEMBL74506 0.72 PDE4A (0.46) ALDH1A1KDM4ELMNAPOLBPKM
SCHEMBL29164216 0.72 ALDH1A1 (0.47) CFTRALDH1A1HPGDHSD17B10CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023000834-A1 BENZIMIDAZOLE OR AZABENZIMIDAZOLE-6-CARBOXYLIC ACID COMPOUND AND USE THEREOF 广州必贝特医药股份有限公司 2023-01-26 WO disclosed
CN-113480534-B Benzimidazole or azabenzimidazole-6-carboxylic acid compounds and application thereof 广州必贝特医药股份有限公司 2022-05-13 CN disclosed
CN-113480534-A Benzimidazole or azabenzimidazole-6-carboxylic acid compounds and application thereof 广州必贝特医药技术有限公司 2021-10-08 CN disclosed