SCHEMBL2494735

SCHEMBL2494735

N=c1n(CCCOc2ccc(Cl)cc2Cl)c2ccccc2n1Cc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.66
MAPT P10636 4/20 0.66
NPSR1 Q6W5P4 3/20 0.66
TSHR P16473 2/20 0.66
MAPK1 P28482 2/20 0.66
LMNA P02545 6/20 0.65
SMN1; SMN2 Q16637 4/20 0.65
KMT2A Q03164 3/20 0.65
XBP1 P17861 2/20 0.65
MEN1 O00255 1/20 0.65
GAA P10253 1/20 0.65
IDE P14735 1/20 0.65
PAX8 Q06710 1/20 0.65
SLC5A2 P31639 2/20 0.51
ALDH1A1 P00352 1/20 0.50
F8 P00451 1/20 0.49
F5 P12259 1/20 0.49
NPC1 O15118 1/20 0.48
PKM P14618 1/20 0.48
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17761715 0.92 TP53 (0.65) TP53MAPTNPSR1TSHRMAPK1
SCHEMBL17761818 0.87 TP53 (0.67) TP53MAPTNPSR1TSHRMAPK1
SCHEMBL17749511 0.87 TP53 (0.67) TP53MAPTNPSR1TSHRMAPK1
SCHEMBL17761637 0.84 TP53 (0.53) TP53MAPTNPSR1TSHRMAPK1
SCHEMBL17761822 0.84 TP53 (0.64) TP53MAPTNPSR1TSHRMAPK1
SCHEMBL17749525 0.83 TP53 (0.60) TP53MAPTNPSR1TSHRMAPK1
SCHEMBL17749595 0.83 SMN1; SMN2 (0.70) TP53MAPTNPSR1TSHRMAPK1
SCHEMBL17761820 0.83 TP53 (0.62) TP53MAPTNPSR1TSHRMAPK1
SCHEMBL17749535 0.82 TP53 (0.71) TP53MAPTNPSR1TSHRMAPK1
SCHEMBL17749548 0.82 TP53 (0.64) TP53MAPTNPSR1TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373629-A1 COMPOUNDS FOR TREATING CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-10-12 EP disclosed
WO-2010067067-A1 COMPOUNDS FOR TREATING CANCER EVOTEC AG (DE) 2010-06-17 WO disclosed