SCHEMBL24947656

SCHEMBL24947656

CCOC(COc1cccc(C)c1F)OCC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.38
KDM4E B2RXH2 1/20 0.38
SCN4A P35499 5/20 0.37
ALOX15 P16050 1/20 0.36
LMNA P02545 3/20 0.34
SCN1A P35498 2/20 0.34
SCN5A Q14524 2/20 0.34
SCN9A Q15858 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
KCNK3 O14649 1/20 0.34
CACNA1F O60840 1/20 0.34
KCNK2 O95069 1/20 0.34
GBA1 P04062 1/20 0.34
MAOA P21397 1/20 0.34
HTR2A P28223 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4551683 0.83 KDM4E (0.54) CYP1A2KDM4ESCN4AALOX15LMNA
SCHEMBL16048103 0.83 KMT2A (0.35) CYP1A2ALOX15CYP2D6MEN1KMT2A
SCHEMBL256772 0.81 L3MBTL1 (0.47) CYP1A2KDM4ELMNACYP2D6MEN1
SCHEMBL18305182 0.81 CYP1A2 (0.38) CYP1A2KDM4ESCN4AALOX15LMNA
SCHEMBL29678765 0.81 CYP1A2 (0.38) CYP1A2KDM4ESCN4AALOX15LMNA
SCHEMBL249260 0.78 L3MBTL1 (0.54) CYP1A2KDM4EALOX15LMNACYP2D6
SCHEMBL9340479 0.78 SCN4A (0.56) CYP1A2SCN4ALMNASCN1ASCN5A
SCHEMBL29559341 0.77 FFAR1 (0.42) CYP1A2KDM4ESCN4AALOX15LMNA
SCHEMBL5987150 0.76 L3MBTL1 (0.38) CYP1A2KDM4EALOX15CYP2D6MEN1
SCHEMBL8534037 0.76 CYP1A2 (0.35) CYP1A2KDM4ELMNASCN1ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023000834-A1 BENZIMIDAZOLE OR AZABENZIMIDAZOLE-6-CARBOXYLIC ACID COMPOUND AND USE THEREOF 广州必贝特医药股份有限公司 2023-01-26 WO disclosed
WO-2023000834-A1 BENZIMIDAZOLE OR AZABENZIMIDAZOLE-6-CARBOXYLIC ACID COMPOUND AND USE THEREOF 广州必贝特医药股份有限公司 2023-01-26 WO disclosed
CN-113480534-B Benzimidazole or azabenzimidazole-6-carboxylic acid compounds and application thereof 广州必贝特医药股份有限公司 2022-05-13 CN disclosed
CN-113480534-A Benzimidazole or azabenzimidazole-6-carboxylic acid compounds and application thereof 广州必贝特医药技术有限公司 2021-10-08 CN disclosed