SCHEMBL24968217

SCHEMBL24968217

COc1ncc(C2CCCC2CO)cc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 11/20 0.35
PIK3CA P42336 10/20 0.35
PIK3CB P42338 2/20 0.33
SSTR4 P31391 2/20 0.32
HTR2B P41595 1/20 0.32
PIK3CG P48736 1/20 0.32
PRKDC P78527 1/20 0.32
PDE4D Q08499 1/20 0.32
AURKA O14965 1/20 0.32
KDR P35968 1/20 0.32
AURKB Q96GD4 1/20 0.32
PIK3R1 P27986 1/20 0.32
RIPK1 Q13546 1/20 0.32
KCNK3 O14649 1/20 0.31
FFAR1 O14842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30851325 1.00 PIK3CD (0.35) PIK3CDPIK3CAPIK3CBSSTR4HTR2B
SCHEMBL27233804 0.84 AR (0.45) PIK3CDPIK3CAPIK3CBAURKAKDR
SCHEMBL27233739 0.84 AR (0.45) PIK3CDPIK3CAPIK3CBAURKAKDR
SCHEMBL27233810 0.84 AR (0.45) PIK3CDPIK3CAPIK3CBAURKAKDR
SCHEMBL24968932 0.84 AR (0.45) PIK3CDPIK3CAPIK3CBAURKAKDR
SCHEMBL24968340 0.84 AR (0.45) PIK3CDPIK3CAPIK3CBAURKAKDR
SCHEMBL24968337 0.84 AR (0.45) PIK3CDPIK3CAPIK3CBAURKAKDR
SCHEMBL24968215 0.82 FFAR1 (0.35) PIK3CDPIK3CAPIK3CBSSTR4RIPK1
SCHEMBL24968213 0.79 SLC6A2 (0.44) PIK3CDPIK3CAPIK3CBSSTR4HTR2B
SCHEMBL24968383 0.78 TACR1 (0.35) PIK3CDPIK3CAPIK3CBSSTR4HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4378938-A1 NOVEL PARP7 INHIBITOR AND USE THEREOF Shanghai Qilu Pharmaceutical Research and Development Centre Ltd. (CN) 2024-06-05 EP disclosed
CN-117642393-A Novel PARP7 inhibitor and application thereof 上海齐鲁制药研究中心有限公司 2024-03-01 CN disclosed
WO-2023006013-A1 NOVEL PARP7 INHIBITOR AND USE THEREOF 上海齐鲁制药研究中心有限公司 2023-02-02 WO disclosed