SCHEMBL24968243

SCHEMBL24968243

Cc1ncc2c(=O)[nH]ccn12

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 16/20 0.45
TNKS O95271 2/20 0.41
PARP1 P09874 2/20 0.41
TNKS2 Q9H2K2 2/20 0.41
PDPK1 O15530 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24968165 0.77 PDE9A (0.39) BRD4
SCHEMBL18185706 0.75 PDE1A (0.43) BRD4
SCHEMBL13522607 0.74 MAPK1 (0.33) BRD4
SCHEMBL1874812 0.73 MEN1 (0.47) BRD4TNKSPARP1TNKS2PDPK1
SCHEMBL18185760 0.73 PDE1C (0.49)
SCHEMBL24859515 0.70 BRD4 (0.41) BRD4
SCHEMBL18519546 0.68 ADORA3 (0.44) BRD4
SCHEMBL22828057 0.68 PDE1B (0.36) TNKSPARP1TNKS2
SCHEMBL18956004 0.68 BRD4 (0.54) BRD4PDPK1
SCHEMBL18185696 0.67 PDE1B (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119894897-A Heteroaromatic compounds for the treatment of neurological disorders 苏文生命科学有限公司 2025-04-25 CN disclosed
US-12162890-B2 Heteroaromatic NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2024-12-10 US disclosed
WO-2023006013-A1 NOVEL PARP7 INHIBITOR AND USE THEREOF 上海齐鲁制药研究中心有限公司 2023-02-02 WO disclosed
US-20230023543-A1 HETEROAROMATIC NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2023-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12162890-B2 Heteroaromatic NMDA receptor modulators and uses thereof GRIN2C, GRIN2A, GRIN1 BRD4 1947/4885TNKS 2608/4885PARP1 3415/4885
US-20230023543-A1 HETEROAROMATIC NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN2C, GRIN2A, GRIN1 BRD4 1947/4885TNKS 2608/4885PARP1 3415/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.