SCHEMBL2496830

SCHEMBL2496830

NS(=O)(=O)c1ccc(CCNC(=O)CC[C@H](NC(=O)NC(CCCCN(Cc2nccn2CC(=O)O)Cc2nccn2CC(=O)O)C(=O)O)C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA1 P00915 14/20 0.46
CA2 P00918 14/20 0.46
CA12 O43570 5/20 0.46
CA9 Q16790 5/20 0.46
CA4 P22748 5/20 0.42
FOLH1 Q04609 5/20 0.42
HSD17B10 Q99714 1/20 0.41
CA5A P35218 2/20 0.40
CA7 P43166 2/20 0.40
CA14 Q9ULX7 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2496817 1.00 CA1 (0.46) CA1CA2CA12CA9CA4
SCHEMBL2835696 0.85 CA2 (0.45) CA1CA2CA12CA9HSD17B10
SCHEMBL2835690 0.85 CA2 (0.45) CA1CA2CA12CA9HSD17B10
SCHEMBL2835689 0.85 CA2 (0.45) CA1CA2CA12CA9HSD17B10
SCHEMBL10292503 0.84 CA2 (0.47) CA1CA2FOLH1
SCHEMBL17997541 0.82 FOLH1 (0.52) FOLH1
SCHEMBL15512642 0.82 FOLH1 (0.52) FOLH1
SCHEMBL2794828 0.82 FOLH1 (0.52) FOLH1
SCHEMBL23553141 0.82 FOLH1 (0.47) FOLH1
SCHEMBL22984221 0.82 FOLH1 (0.47) FOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373621-A2 TECHNETIUM-AND RHENIUM-BIS(HETEROARYL)COMPLEXES AND METHODS OF USE THEREOF Molecular Insight Pharmaceuticals, Inc. (US) 2011-10-12 EP disclosed
WO-2010065899-A2 TECHNETIUM-AND RHENIUM-BIS(HETEROARYL)COMPLEXES AND METHODS OF USE THEREOF MOLECULAR INSIGHT PHARMACEUTICALS, INC. (US) 2010-06-10 WO disclosed