SCHEMBL24969725

SCHEMBL24969725

CC(C)(C)OC(=O)NCCc1ccccc1C#Cc1cnc(N2CCN(C(=O)OC(C)(C)C)CC2)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.46
P2RY12 Q9H244 4/20 0.42
NR1H2 P55055 1/20 0.42
NR1H3 Q13133 1/20 0.42
SLC2A1 P11166 3/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CKS1B P61024 1/20 0.40
SKP1 P63208 1/20 0.40
SKP2 Q13309 1/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
ADK P55263 1/20 0.39
ACHE P22303 1/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
CXCR3 P49682 1/20 0.38
CCNK O75909 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31142967 1.00 KIT (0.46) KITP2RY12NR1H2NR1H3SLC2A1
SCHEMBL31142973 0.87 P2RY12 (0.46) KITP2RY12NR1H2NR1H3MEN1
SCHEMBL24969726 0.86 P2RY12 (0.46) KITP2RY12NR1H2NR1H3MEN1
SCHEMBL31143040 0.83 MEN1 (0.44) KITP2RY12NR1H2NR1H3MEN1
SCHEMBL31143082 0.82 MEN1 (0.46) KITNR1H2NR1H3MEN1KMT2A
SCHEMBL31143001 0.82 MEN1 (0.43) KITNR1H2NR1H3MEN1KMT2A
SCHEMBL19212401 0.76 P2RY12 (0.54) KITP2RY12SLC2A1MEN1KMT2A
SCHEMBL31142861 0.75 MEN1 (0.47) KITNR1H2NR1H3MEN1KMT2A
SCHEMBL31142932 0.75 NR1H2 (0.43) KITP2RY12NR1H2NR1H3MEN1
SCHEMBL24969739 0.74 SMN1; SMN2 (0.48) P2RY12MEN1KMT2ALMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002011-A1 GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-01-26 WO disclosed