SCHEMBL24975308

SCHEMBL24975308

Cc1cnc(CN(C)CC2Cc3c(cccc3N3CCCCC3)CN2)c(C)c1

nearest known ligand 0.85

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 20/20 0.85
CYP2D6 P10635 11/20 0.85
CHRM2 P08172 8/20 0.85
CHRM4 P08173 8/20 0.85
CHRM5 P08912 8/20 0.85
CHRM1 P11229 8/20 0.85
CHRM3 P20309 8/20 0.85
CYP3A4 P08684 4/20 0.65
KCNH2 Q12809 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20483199 0.92 CXCR4 (1.00) CXCR4CYP2D6CHRM2CHRM4CHRM5
SCHEMBL20483202 0.92 CXCR4 (1.00) CXCR4CYP2D6CHRM2CHRM4CHRM5
SCHEMBL21744551 0.91 CXCR4 (0.82) CXCR4CYP2D6CHRM2CHRM4CHRM5
SCHEMBL21743938 0.91 CXCR4 (0.82) CXCR4CYP2D6CHRM2CHRM4CHRM5
SCHEMBL21744836 0.91 CXCR4 (0.82) CXCR4CYP2D6CHRM2CHRM4CHRM5
SCHEMBL21744151 0.90 CXCR4 (0.81) CXCR4CYP2D6CHRM2CHRM4CHRM5
SCHEMBL21744546 0.89 CXCR4 (0.79) CXCR4CYP2D6CHRM2CHRM4CHRM5
SCHEMBL21743754 0.87 CXCR4 (0.72) CXCR4CYP2D6CHRM2CHRM4CHRM5
SCHEMBL30239422 0.82 CXCR4 (0.69) CXCR4CYP2D6CHRM2CHRM4CHRM5
SCHEMBL20483201 0.79 CXCR4 (1.00) CXCR4CYP2D6CHRM2CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023003862-A1 CXCR4 MODULATORS AND USES RELATED THERETO EMORY UNIVERSITY (US) 2023-01-26 WO disclosed