SCHEMBL24975663

SCHEMBL24975663

COc1ccn2c(-c3cncc(N[C@H]4CNC[C@@H]4F)n3)cnc2c1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 9/20 0.62
IRAK4 Q9NWZ3 3/20 0.44
KDR P35968 5/20 0.43
KIT P10721 5/20 0.43
CSF1R P07333 4/20 0.43
CYP2D6 P10635 1/20 0.43
KCNH2 Q12809 1/20 0.43
DYRK1A Q13627 3/20 0.41
CLK2 P49760 2/20 0.41
CLK3 P49761 2/20 0.41
NRAS P01111 1/20 0.39
GSK3B P49841 1/20 0.39
IGF1R P08069 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24977141 0.92 FLT3 (0.57) FLT3IRAK4KDRKITCSF1R
SCHEMBL27362520 0.92 FLT3 (0.57) FLT3IRAK4KDRKITCSF1R
SCHEMBL24231493 0.91 FLT3 (0.52) FLT3IRAK4KDRKITCSF1R
SCHEMBL24975664 0.90 FLT3 (0.50) FLT3IRAK4KDRKITCSF1R
SCHEMBL24975661 0.90 FLT3 (0.50) FLT3IRAK4KDRKITCSF1R
SCHEMBL25989696 0.89 FLT3 (0.79) FLT3IRAK4KDRKITCSF1R
SCHEMBL25989694 0.89 FLT3 (0.79) FLT3IRAK4KDRKITCSF1R
SCHEMBL24231529 0.89 FLT3 (0.79) FLT3IRAK4KDRKITCSF1R
SCHEMBL24975668 0.88 FLT3 (0.49) FLT3IRAK4KDRKITCSF1R
SCHEMBL10239879 0.87 FLT3 (0.60) FLT3IRAK4KDRKITCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250154144-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF CHILDRENS HOSPITAL MED CT (US) 2025-05-15 US disclosed
WO-2023009833-A9 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2023-11-23 WO disclosed
WO-2023009833-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2023-02-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250154144-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF FLT3, IRAK1, IRAK3 FLT3 1/4885IRAK4 5/4885KDR 737/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.