SCHEMBL24975833

SCHEMBL24975833

Cc1nc(-c2cnn(C)c2)c2ccccc2n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.49
EPHX2 P34913 1/20 0.48
AXL P30530 4/20 0.46
BRD4 O60885 1/20 0.46
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 3/20 0.45
HTT P42858 2/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HSD17B10 Q99714 1/20 0.45
KDM1A O60341 1/20 0.44
GRM4 Q14833 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PIM1 P11309 1/20 0.41
ADORA2A P29274 1/20 0.41
PFKFB3 Q16875 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NUDT1 P36639 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31428805 1.00 GRM2 (0.49) GRM2EPHX2AXLBRD4KDM4E
SCHEMBL31428997 0.80 GRM2 (0.51) GRM2EPHX2AXLBRD4KDM4E
SCHEMBL1773091 0.78 NUDT1 (0.60) KDM4EALDH1A1HTTMAPTHPGD
SCHEMBL31428664 0.77 GRM4 (0.65) GRM2EPHX2AXLBRD4GRM4
SCHEMBL17942808 0.76 AXL (0.49) GRM2EPHX2AXLBRD4KDM1A
SCHEMBL29986553 0.75 ADORA2A (0.57) KDM4EALDH1A1HTTMAPTHPGD
SCHEMBL16542819 0.75 ADORA2A (0.57) KDM4EALDH1A1HTTMAPTHPGD
SCHEMBL17942680 0.75 BRD4 (0.44) GRM2EPHX2AXLBRD4MAPT
SCHEMBL31429051 0.75 GRM2 (0.64) GRM2EPHX2BRD4KDM4EALDH1A1
SCHEMBL24977215 0.75 GRM2 (0.64) GRM2EPHX2BRD4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023008577-A1 RAS/RAF BINDING INHIBITOR COMPOUND 国立大学法人神戸大学 2023-02-02 WO disclosed