SCHEMBL25003385

SCHEMBL25003385

Cc1ccc(CNC(=O)c2cc3ccccc3s2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 5/20 0.66
HDAC1 Q13547 5/20 0.66
HDAC3 O15379 2/20 0.66
NCOR2 Q9Y618 1/20 0.66
OPRM1 P35372 4/20 0.62
OPRD1 P41143 1/20 0.62
OPRL1 P41146 1/20 0.62
RAB9A P51151 1/20 0.60
CLK1 P49759 1/20 0.59
SENP5 Q96HI0 1/20 0.59
SENP2 Q9HC62 1/20 0.59
SENP1 Q9P0U3 1/20 0.59
HDAC4 P56524 1/20 0.57
HDAC7 Q8WUI4 1/20 0.57
HDAC10 Q969S8 1/20 0.57
HDAC11 Q96DB2 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
HDAC9 Q9UKV0 1/20 0.57
HDAC5 Q9UQL6 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29617711 0.84 HDAC2 (0.60) HDAC2HDAC1HDAC3NCOR2RAB9A
SCHEMBL6919078 0.84 HDAC1 (0.70) HDAC2HDAC1HDAC3NCOR2RAB9A
SCHEMBL18641949 0.84 HDAC2 (0.60) HDAC2HDAC1HDAC3NCOR2RAB9A
SCHEMBL28863161 0.84 HDAC1 (0.60) HDAC2HDAC1HDAC3NCOR2OPRM1
SCHEMBL12057508 0.82 HDAC2 (0.67) HDAC2HDAC1HDAC3NCOR2RAB9A
SCHEMBL13494017 0.82 HDAC2 (0.63) HDAC2HDAC1HDAC3NCOR2RAB9A
SCHEMBL15246624 0.82 NAMPT (0.69) HDAC2HDAC1HDAC3NCOR2NAMPT
SCHEMBL16141033 0.81 CLK1 (0.56) HDAC2HDAC1HDAC3NCOR2RAB9A
SCHEMBL16142440 0.80 PPARA (0.53) HDAC2HDAC1HDAC3NCOR2CLK1
SCHEMBL30180461 0.80 HDAC2 (1.00) HDAC2HDAC1HDAC3NCOR2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011416-A1 MULTI-TARGET INHIBITOR TARGETING HDAC AND NAD SYNTHESIS AND USE OF MULTI-TARGET INHIBITOR 中国海洋大学 2023-02-09 WO disclosed