SCHEMBL25003553

SCHEMBL25003553

O=Cc1ccc(CNC(=O)c2cc3cnccc3[nH]2)cc1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 19/20 0.69
CYP2C9 P11712 5/20 0.69
HDAC1 Q13547 2/20 0.63
HDAC3 O15379 1/20 0.63
HDAC2 Q92769 1/20 0.63
NCOR2 Q9Y618 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15246211 0.86 NAMPT (0.76) NAMPTCYP2C9HDAC1HDAC3HDAC2
SCHEMBL28954653 0.85 NAMPT (0.78) NAMPTCYP2C9HDAC1HDAC3HDAC2
SCHEMBL1647859 0.82 NAMPT (0.71) NAMPTCYP2C9HDAC1HDAC3HDAC2
SCHEMBL25002581 0.82 NAMPT (1.00) NAMPTCYP2C9HDAC1HDAC3HDAC2
SCHEMBL160706 0.80 NAMPT (1.00) NAMPTCYP2C9
SCHEMBL25002551 0.80 HDAC2 (0.62) HDAC1HDAC3HDAC2
SCHEMBL25002623 0.80 NHERF1 (0.76) HDAC1HDAC3HDAC2
SCHEMBL168504 0.79 NAMPT (0.83) NAMPTCYP2C9
SCHEMBL12468236 0.79 NAMPT (0.84) NAMPTCYP2C9
SCHEMBL16107639 0.79 HDAC1 (0.72) NAMPTCYP2C9HDAC1HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011416-A1 MULTI-TARGET INHIBITOR TARGETING HDAC AND NAD SYNTHESIS AND USE OF MULTI-TARGET INHIBITOR 中国海洋大学 2023-02-09 WO disclosed