SCHEMBL25020191

SCHEMBL25020191

CC(N)c1cccc(CC(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
TAAR1 Q96RJ0 4/20 0.38
SLC6A2 P23975 2/20 0.38
MAOA P21397 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
CYP2A6 P11509 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
PDE2A O00408 1/20 0.37
PNMT P11086 1/20 0.37
TACR1 P25103 1/20 0.36
CFD P00746 1/20 0.35
F11 P03951 1/20 0.35
TPSB2 P20231 1/20 0.35
KRAS P01116 1/20 0.35
SOS1 Q07889 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21133179 1.00 HTR2A (0.45) HTR2AHTR2CHTR2BTAAR1SLC6A2
SCHEMBL14120621 0.85 PTPN5 (0.43) HTR2AHTR2CHTR2BSLC6A4SIGMAR1
SCHEMBL18266583 0.85 HTR2A (0.41) HTR2AHTR2CHTR2BTAAR1SLC6A2
SCHEMBL14259225 0.82 HTR2A (0.41) HTR2AHTR2CHTR2BTAAR1SLC6A4
SCHEMBL11414162 0.80 HTR2A (0.64) HTR2AHTR2CHTR2BTAAR1SLC6A2
SCHEMBL28644938 0.79 TAAR1 (0.42) HTR2AHTR2CHTR2BTAAR1SLC6A2
SCHEMBL20431924 0.78 SLC22A1 (0.37) HTR2AHTR2CHTR2BTAAR1SLC6A2
SCHEMBL24324366 0.78 TAAR1 (0.41) TAAR1SLC6A2MAOASLC6A4SLC6A3
SCHEMBL29342899 0.77 TAAR1 (0.43) HTR2AHTR2CHTR2BTAAR1SLC6A2
SCHEMBL28856242 0.77 PNMT (0.47) TAAR1SLC6A2MAOASLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3728254-B1 BENZYLAMINO SUBSTITUTED PYRIDOPYRIMIDINONES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2023-02-15 EP disclosed