SCHEMBL25045802

SCHEMBL25045802

Cc1cnn2c(I)cccc12

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40
CYP17A1 P05093 1/20 0.35
CYP1A2 P05177 1/20 0.35
TLR8 Q9NR97 1/20 0.32
KDM4E B2RXH2 1/20 0.31
HTT P42858 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25044269 0.79 DRD2 (0.41) DRD2DRD4DRD3
SCHEMBL21863437 0.79 DRD2 (0.41) DRD2DRD4DRD3CYP17A1CYP1A2
SCHEMBL24103795 0.76 TSHR (0.36) CYP17A1CYP1A2TLR8KDM4EHTT
SCHEMBL12145712 0.74 DRD4 (0.41) DRD4DRD3CYP17A1CYP1A2HTT
SCHEMBL23938203 0.73 CYP17A1 (0.33) DRD2DRD4DRD3CYP17A1CYP1A2
SCHEMBL21893906 0.73 PDE4B (0.33) CYP17A1CYP1A2TLR8NPC1RAB9A
SCHEMBL5848633 0.72 DRD2 (0.38) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL23938202 0.72 CYP1A2 (0.35) CYP17A1CYP1A2TLR8
SCHEMBL24729869 0.68 DRD2 (0.40) DRD2DRD4DRD3CYP17A1CYP1A2
SCHEMBL21631042 0.67 IDO1 (0.41) DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230050653-A1 ROCK INHIBITOR AND PREPARATION METHOD THEREFOR AND USE THEREOF WUHAN LL SCIENCE AND TECHNOLOGY DEVELOPMENT CO., LTD. (CN) 2023-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230050653-A1 ROCK INHIBITOR AND PREPARATION METHOD THEREFOR AND USE THEREOF ROCK1, CYP11B1, CYP4A11 DRD2 3504/4885DRD4 3371/4885DRD3 3447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.