SCHEMBL25057796

SCHEMBL25057796

Nc1nc(N2CCC(c3nnc4n3-c3ccc(Cl)cc3CN(CC3(F)COC3)C4)CC2)ccc1F

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 10/20 0.47
AVPR1A P37288 12/20 0.47
KCNH2 Q12809 4/20 0.47
OXTR P30559 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20728257 0.91 OXTR (0.57) AVPR2AVPR1AKCNH2OXTR
SCHEMBL20727970 0.90 AVPR2 (0.47) AVPR2AVPR1AKCNH2OXTR
SCHEMBL20728117 0.90 AVPR2 (0.46) AVPR2AVPR1AKCNH2OXTR
SCHEMBL20728115 0.90 AVPR2 (0.46) AVPR2AVPR1AKCNH2OXTR
SCHEMBL20728265 0.88 AVPR2 (0.62) AVPR2AVPR1AKCNH2OXTR
SCHEMBL20728280 0.87 AVPR1A (0.49) AVPR2AVPR1AKCNH2OXTR
SCHEMBL20728269 0.86 AVPR1A (0.53) AVPR2AVPR1AKCNH2OXTR
SCHEMBL20728500 0.86 AVPR1A (0.57) AVPR2AVPR1AKCNH2OXTR
SCHEMBL20728454 0.85 AVPR1A (0.46) AVPR2AVPR1AKCNH2OXTR
SCHEMBL20727943 0.85 AVPR2 (0.51) AVPR2AVPR1AKCNH2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3634963-B1 1-(2-AZASPIRO[3.3]HEPTAN-6-YL)-5,6-DIHYDRO-4H-BENZO[F][1,2,4]TRIAZOLO[4,3-A][1,4]DIAZEPINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS FOR TREATING NEUROPSYCHOLOGICAL DISORDERS BLACKTHORN THERAPEUTICS INC (US) 2023-02-22 EP disclosed