SCHEMBL250602

SCHEMBL250602

C1=Cc2nc3ccccc3cc2OC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
MAPT P10636 5/20 0.42
HPGD P15428 5/20 0.42
GLA P06280 3/20 0.42
ACHE P22303 1/20 0.42
KDM4E B2RXH2 6/20 0.37
KMT2A Q03164 5/20 0.37
NPC1 O15118 4/20 0.37
RAB9A P51151 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
MEN1 O00255 3/20 0.37
TP53 P04637 3/20 0.37
PKM P14618 3/20 0.37
HSD17B10 Q99714 3/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
TSHR P16473 2/20 0.37
MAPK1 P28482 2/20 0.37
CYP2C19 P33261 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Indoline SCHEMBL9236550 0.83 MEN1 (0.33) ALDH1A1MAPTHPGDACHEKDM4E
Acridine SCHEMBL28072004 0.77 MAPT (0.48) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL28360837 0.74 HPRT1 (0.39) ALDH1A1MAPTHPGDGLAKDM4E
SCHEMBL1040670 0.72 ALDH1A1 (0.42) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL30536492 0.71 STS (0.45) CYP1A2POLBCYP1A1
SCHEMBL3033164 0.71 STS (0.45) CYP1A2POLBCYP1A1
SCHEMBL5177973 0.69 ALDH1A1 (0.46) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL30530594 0.69 ALDH1A1 (0.42) ALDH1A1MAPTHPGDGLAACHE
Iodide SCHEMBL3900318 0.68 ALDH1A1 (0.45) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL28430609 0.68 ALDH1A1 (0.45) ALDH1A1MAPTHPGDGLAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 539 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4304842-B1 METHOD FOR MAKING PHOTOFUNCTIONAL CONTACT LENSES ALCON INC (CH) 2026-05-06 EP claimed
US-12285922-B2 Method for making photofunctional contact lenses ALCON INC. (CH) 2025-04-29 US claimed
US-12247169-B2 Method for making photochromic contact lenses ALCON INC. (CH) 2025-03-11 US claimed
EP-4514597-A1 METHOD FOR MAKING UV AND HEVL-ABSORBING OPHTHALMIC LENSES Alcon Inc. (CH) 2025-03-05 EP claimed
EP-4313567-B1 METHOD FOR MAKING PHOTOCHROMIC CONTACT LENSES ALCON INC (CH) 2025-01-29 EP claimed
EP-4237232-B1 METHOD FOR MAKING PHOTOCHROMIC CONTACT LENSES ALCON INC (CH) 2024-11-27 EP claimed
US-12111443-B2 Method for making photochromic contact lenses ALCON INC. (CH) 2024-10-08 US claimed
US-20240287379-A1 METHOD FOR MAKING PHOTOCHROMIC CONTACT LENSES ALCON INC. (CH) 2024-08-29 US claimed
US-11999908-B2 Method for making photochromic contact lenses ALCON INC. (CH) 2024-06-04 US claimed
EP-2718755-B1 POLARIZING PHOTOCHROMIC ARTICLES TRANSITIONS OPTICAL INC (US) 2024-05-29 EP claimed
US-20060022176-A1 Reaction product of a ring-opening cyclic ester or carbonate and a photochromic initiator, especially a naphtho[1,2-b]quinone with one or more hydroxy groups, e.g., (1) 3,3-di(4-methoxyphenyl)-6,7-dimethoxy-13-methyl-13-(2-(2-hydroxyethoxy)ethoxy)-3H,13H-indeno[2,1-f]naphtho[1,2-b]pyran. TRANSITIONS OPTICAL LIMITED (IE) 2006-02-02 US claimed
CN-1729266-A Photochromic compositions and light transmissible articles POLYMERS AUSTRALIA PTY LTD (AU) 2006-02-01 CN claimed
EP-1037951-B1 PHOTOCHROMIC EPOXY RESIN COATING COMPOSITION PPG IND OHIO INC (US) 2005-11-16 EP claimed
EP-1149138-B1 POLYANHYDRIDE PHOTOCHROMIC COATING COMPOSITION AND PHOTOCHROMIC ARTICLES PPG IND OHIO INC (US) 2005-03-09 EP claimed
EP-1230232-B1 SUBSTITUTED 4H-CHROMENE AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA INC (US) 2004-02-25 EP claimed
EP-1230232-A2 SUBSTITUTED 4H-CHROMENE AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF Cytovia, Inc. (US) 2002-08-14 EP claimed
US-6268055-B1 CURED OVERCOATING PPG INDUSTRIES OHIO, INC. 2001-07-31 US claimed
WO-2001034591-A2 SUBSTITUTED 4H-CHROMENE AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2001-05-17 WO claimed
EP-1037951-A1 PHOTOCHROMIC EPOXY RESIN COATING COMPOSITION PPG Industries Ohio, Inc. (US) 2000-09-27 EP claimed
WO-1999029791-A1 PHOTOCHROMIC EPOXY RESIN COATING COMPOSITION PPG INDUSTRIES OHIO, INC. (US) 1999-06-17 WO claimed