SCHEMBL25072096

SCHEMBL25072096

CC(C)(C)OC(=O)N[C@H]1CC[C@H](Nc2nccc(-c3cccnc3Oc3c(F)cc(N)cc3Cl)n2)CC1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 19/20 0.48
MAPK10 P53779 10/20 0.48
KDR P35968 1/20 0.38
TEK Q02763 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28551474 1.00 ERN1 (0.48) ERN1MAPK10KDRTEK
SCHEMBL21908731 1.00 ERN1 (0.48) ERN1MAPK10KDRTEK
SCHEMBL21909261 0.95 ERN1 (0.46) ERN1MAPK10
SCHEMBL25071801 0.95 ERN1 (0.46) ERN1MAPK10
SCHEMBL28554822 0.95 ERN1 (0.46) ERN1MAPK10
SCHEMBL28555901 0.92 ERN1 (0.49) ERN1MAPK10
SCHEMBL25071795 0.92 ERN1 (0.49) ERN1MAPK10
SCHEMBL25071948 0.86 ERN1 (0.57) ERN1MAPK10
SCHEMBL21811392 0.86 ERN1 (0.57) ERN1MAPK10
SCHEMBL30143179 0.86 ERN1 (0.57) ERN1MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230057166-A1 PHENOXY-PYRIDYL-PYRIMIDINE COMPOUNDS AND METHODS OF USE GENENTECH INC (US) 2023-02-23 US disclosed
CN-112739420-A Phenoxy-pyridyl-pyrimidine compounds and methods of use 基因泰克公司 2021-04-30 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230057166-A1 PHENOXY-PYRIDYL-PYRIMIDINE COMPOUNDS AND METHODS OF USE XBP1, ERN1, ESR2 ERN1 2/4885MAPK10 1353/4885KDR 2456/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.