SCHEMBL25091099

SCHEMBL25091099

CCC1CCN(C(=O)c2ccc(-c3cn(C)c(=O)c(C)c3C)cc2OC(F)(F)F)C2(CC2)C1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.35
CYP3A4 P08684 1/20 0.34
BRD4 O60885 2/20 0.33
BRD2 P25440 1/20 0.33
BRD9 Q9H8M2 1/20 0.33
BRD7 Q9NPI1 1/20 0.33
HCRTR1 O43613 2/20 0.32
HCRTR2 O43614 2/20 0.32
PIK3CA P42336 6/20 0.32
MTOR P42345 6/20 0.32
SSTR4 P31391 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23798067 0.89 CACNA1B (0.35) CACNA1BCYP3A4BRD4BRD2BRD9
SCHEMBL25844139 0.79 BRD9 (0.39) CYP3A4BRD4BRD2BRD9BRD7
SCHEMBL25091781 0.77 CACNA1B (0.45) CACNA1BCYP3A4BRD4BRD2BRD9
SCHEMBL23798059 0.75 CACNA1B (0.38) CACNA1BCYP3A4BRD4BRD2BRD9
SCHEMBL25091954 0.75 BRD4 (0.38) BRD4BRD2BRD9BRD7
SCHEMBL23783402 0.74 BRD4 (0.43) BRD4BRD2BRD9BRD7
SCHEMBL30031484 0.74 BRD4 (0.43) BRD4BRD2BRD9BRD7
SCHEMBL23783182 0.74 BRD4 (0.43) BRD4BRD2BRD9BRD7
SCHEMBL25091776 0.72 CACNA1B (0.44) CACNA1BCYP3A4BRD4BRD9PIK3CA
SCHEMBL25091093 0.71 METAP2 (0.43) CACNA1BCYP3A4BRD4BRD9PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230060334-A1 COMPOUNDS FOR TARGETED DEGRADATION OF BRD9 C4 THERAPEUTICS, INC. (US) 2023-03-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230060334-A1 COMPOUNDS FOR TARGETED DEGRADATION OF BRD9 BRD9, BRD1, BRWD1 CACNA1B 4261/4885CYP3A4 4588/4885BRD4 30/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.