SCHEMBL25145641

SCHEMBL25145641

FC(F)(F)c1ccnc(CC2CCNCC2)n1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.48
CACNA1H O95180 2/20 0.46
PIM1 P11309 2/20 0.42
SYK P43405 1/20 0.41
HTR2C P28335 5/20 0.40
HTR2A P28223 4/20 0.40
HTR2B P41595 4/20 0.40
CACNA1G O43497 1/20 0.40
GBA1 P04062 1/20 0.39
MAPK1 P28482 1/20 0.39
PIK3CA P42336 1/20 0.38
KCNH2 Q12809 1/20 0.38
BRD4 O60885 1/20 0.36
HRH4 Q9H3N8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5763019 0.87 ADRB1 (0.45) ADRB1CACNA1HPIM1SYKHTR2C
SCHEMBL31239629 0.79 ADRB1 (0.39) ADRB1CACNA1HSYKHTR2CHTR2A
Hydrochloric Acid SCHEMBL6152965 0.75 HRH4 (0.54) ADRB1PIM1SYKBRD4HRH4
SCHEMBL25145914 0.73 MALT1 (0.43) ADRB1CACNA1HPIM1HTR2CCACNA1G
SCHEMBL5688150 0.73 GBA1 (0.52) CACNA1HGBA1KCNH2HRH4HRH3
SCHEMBL25145546 0.72 CACNA1H (0.47) CACNA1HHTR2CHTR2BCACNA1GGBA1
SCHEMBL25145959 0.72 GBA1 (0.47) CACNA1HCACNA1GGBA1PIK3CAKCNH2
SCHEMBL2243533 0.71 MAPK1 (0.55) ADRB1SYKMAPK1PIK3CAKCNH2
SCHEMBL25145644 0.71 MAPK1 (0.55) ADRB1CACNA1HHTR2CHTR2BCACNA1G
SCHEMBL940757 0.71 SYK (0.51) ADRB1SYKHTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023062049-A1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2023-04-20 WO disclosed