SCHEMBL25147686

SCHEMBL25147686

CNc1cc(Cl)cnc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.43
CHUK O15111 1/20 0.41
PROKR1 Q8TCW9 1/20 0.32
HTT P42858 3/20 0.32
HSD17B10 Q99714 3/20 0.32
IDO1 P14902 1/20 0.32
KAT2B Q92831 1/20 0.32
BRD9 Q9H8M2 1/20 0.32
HPGD P15428 1/20 0.32
JAK2 O60674 1/20 0.31
ALDH1A1 P00352 2/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
LMNA P02545 1/20 0.31
PABPC1 P11940 1/20 0.31
KDM4E B2RXH2 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
FLT1 P17948 1/20 0.31
TRPM5 Q9NZQ8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12393156 0.78 CHUK (0.39) CHUKHTTHSD17B10KAT2BBRD9
SCHEMBL27688260 0.77 NOS3 (0.35) NPC1RAB9ACYP1A2
SCHEMBL7943085 0.77 CHUK (0.38) CHUKPROKR1HTTHSD17B10KAT2B
SCHEMBL3513683 0.75 HTT (0.34) HTTHSD17B10JAK2ALDH1A1KMT2A
SCHEMBL24470415 0.75 CHUK (0.37) CHUKHTTHSD17B10KAT2BBRD9
SCHEMBL20859298 0.75 IDO1 (0.39) CHUKHTTHSD17B10IDO1KAT2B
SCHEMBL28928912 0.72 CYP2C9 (0.43) CHUKMEN1KMT2ALMNATSHR
SCHEMBL27798823 0.72 KCNH2 (0.31) NPC1RAB9A
SCHEMBL635255 0.71
SCHEMBL115615 0.71 PLAU (0.32) GRM4HTTHSD17B10IDO1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064585-A1 7,8-DIHYDRO-5H-1,6-NAPHTHYRIDINE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS VANDERBILT UNIVERSITY (US) 2023-04-20 WO disclosed