SCHEMBL25147753

SCHEMBL25147753

Cc1cc(C#N)nnc1N1CCc2ncc(CC(F)(F)F)cc2C1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.33
PANK3 Q9H999 1/20 0.33
P2RX3 P56373 4/20 0.33
P2RX2 Q9UBL9 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31659520 1.00 KDM4E (0.33) KDM4EPANK3P2RX3P2RX2
SCHEMBL25147761 0.85 P2RX3 (0.35) KDM4EP2RX3P2RX2
SCHEMBL30331940 0.85 P2RX3 (0.35) KDM4EP2RX3P2RX2
SCHEMBL30370412 0.85 KDM4E (0.35) KDM4EP2RX3P2RX2
SCHEMBL25153188 0.85 KDM4E (0.35) KDM4EP2RX3P2RX2
SCHEMBL25148366 0.83 GRIN2D (0.32) KDM4EP2RX3P2RX2
SCHEMBL31659721 0.83 GRIN2D (0.32) KDM4EP2RX3P2RX2
SCHEMBL30332146 0.81 GRIN2D (0.31)
SCHEMBL25148195 0.81 GRIN2D (0.31)
SCHEMBL25147741 0.81 P2RX3 (0.36) P2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064585-A1 7,8-DIHYDRO-5H-1,6-NAPHTHYRIDINE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS VANDERBILT UNIVERSITY (US) 2023-04-20 WO disclosed