SCHEMBL25166014

SCHEMBL25166014

Nc1cc2c(c(Br)c1Cl)OCC2

nearest known ligand 0.36

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25166055 0.90 NOTUM (0.35)
SCHEMBL25166146 0.80 PARP1 (0.37) PARP1
SCHEMBL25166010 0.79 PARP1 (0.42) PARP1
SCHEMBL25166256 0.78 MAPT (0.37)
SCHEMBL30329748 0.72 GPR35 (0.37) PARP1
SCHEMBL30695888 0.72 PARP1 (0.39) PARP1
SCHEMBL4107808 0.72 PARP1 (0.39) PARP1
SCHEMBL4100100 0.72 PARP1 (0.39) PARP1
SCHEMBL30768351 0.72 PARP1 (0.39) PARP1
SCHEMBL24373459 0.71 NOTUM (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118647610-A Novel modulators of EHMT1 and EHMT2 and therapeutic uses thereof 探戈医药股份有限公司 2024-09-13 CN disclosed
EP-4416143-A1 NOVEL MODULATORS OF EHMT1 AND EHMT2 AND THERAPEUTIC USE THEREOF Tango Therapeutics, Inc. (US) 2024-08-21 EP disclosed
WO-2023064586-A1 NOVEL MODULATORS OF EHMT1 AND EHMT2 AND THERAPEUTIC USE THEREOF TANGO THERAPEUTICS, INC. (US) 2023-04-20 WO disclosed
WO-2023064586-A1 NOVEL MODULATORS OF EHMT1 AND EHMT2 AND THERAPEUTIC USE THEREOF TANGO THERAPEUTICS, INC. (US) 2023-04-20 WO disclosed