SCHEMBL25171592

SCHEMBL25171592

c1ccc(CN2CCOC(c3ccccn3)C2)cc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 10/20 0.53
DRD4 P21917 8/20 0.52
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30373788 0.84 DRD4 (0.50) CNR2DRD4CYP1A2CYP3A4CYP2D6
SCHEMBL17888417 0.83 DRD3 (0.51) CNR2DRD4DRD3
SCHEMBL25178173 0.83 CNR2 (0.55) CNR2DRD4CYP1A2CYP3A4CYP2D6
SCHEMBL17224145 0.82 CNR2 (0.49) CNR2DRD4CYP1A2CYP3A4CYP2D6
SCHEMBL26154079 0.82 DRD4 (0.54) CNR2DRD4CYP1A2CYP3A4CYP2D6
SCHEMBL17224143 0.82 CNR2 (0.49) CNR2DRD4CYP1A2CYP3A4CYP2D6
SCHEMBL25184733 0.81 CNR2 (0.50) CNR2DRD4CYP1A2CYP3A4CYP2D6
SCHEMBL4471704 0.80 CNR2 (0.65) CNR2
SCHEMBL14868702 0.80 PDCD1LG2 (0.52) DRD4CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8844465 0.80 PDCD1LG2 (0.52) DRD4CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250051316-A1 2-(ARYL-2-YL) MORPHOLINE AND DEUTERATED DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF SHANGHAI HANSOH BIOMEDICAL CO., LTD. (CN) 2025-02-13 US disclosed
EP-4428128-A1 2-(ARYL-2-YL) MORPHOLINE AND DEUTERATED DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Shanghai Hansoh Biomedical Co., Ltd. (CN) 2024-09-11 EP disclosed
CN-118176185-A 2- (Aryl-2-yl) morpholine and deuterated derivative thereof, preparation method and application 上海翰森生物医药科技有限公司 2024-06-11 CN disclosed
WO-2023078392-A1 2-(ARYL-2-YL) MORPHOLINE AND DEUTERATED DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海翰森生物医药科技有限公司 2023-05-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250051316-A1 2-(ARYL-2-YL) MORPHOLINE AND DEUTERATED DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF TAAR1, TAAR5, AVPR2 CNR2 8/4885DRD4 418/4885CYP1A2 189/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.