SCHEMBL25217836

SCHEMBL25217836

Cc1ccc(C(=O)O)nc1Oc1cccc2cc(OCc3c(-c4c(Cl)cccc4Cl)noc3C3CC3)ccc12

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.59
HSD17B13 Q7Z5P4 1/20 0.56
FABP1 P07148 5/20 0.55
FXR2 P51116 1/20 0.54
FABP4 P15090 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23474151 0.92 NR1H4 (0.63) NR1H4HSD17B13FABP1FXR2FABP4
SCHEMBL23474119 0.89 NR1H4 (0.59) NR1H4HSD17B13FABP1FXR2FABP4
SCHEMBL29726980 0.89 NR1H4 (0.59) NR1H4HSD17B13FABP1FXR2FABP4
SCHEMBL23474095 0.88 NR1H4 (0.59) NR1H4HSD17B13FXR2
SCHEMBL23474194 0.86 NR1H4 (0.58) NR1H4HSD17B13FABP1FXR2FABP4
SCHEMBL23474089 0.85 NR1H4 (0.56) NR1H4HSD17B13FABP1FXR2FABP4
SCHEMBL23474117 0.84 NR1H4 (0.63) NR1H4HSD17B13FXR2
SCHEMBL29726971 0.84 NR1H4 (0.63) NR1H4HSD17B13FXR2
SCHEMBL23474118 0.84 NR1H4 (0.58) NR1H4HSD17B13FABP1FXR2FABP4
SCHEMBL29726969 0.84 NR1H4 (0.58) NR1H4HSD17B13FABP1FXR2FABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4073070-B1 COMPOUNDS FOR MODULATING ACTIVITY OF FXR AND USES THEREOF GANNEX PHARMA CO LTD (CN) 2026-02-18 EP disclosed
US-20230165843-A1 USE AND PHARMACEUTICAL COMPOSITION OF PHENYLISOXAZOLYL METHYLENE-NAPHTHALENE-ETHER DERIVATIVES GANNEX PHARMA CO LTD (CN) 2023-06-01 US disclosed
CN-112898289-B Compounds for modulating FXR activity and uses thereof 甘莱制药有限公司 2022-11-04 CN disclosed
CN-112891348-B Use of phenyl isoxazolyl methylene-naphthalene-ether derivatives and pharmaceutical compositions 甘莱制药有限公司 2022-06-28 CN disclosed
CN-112891348-A Use and pharmaceutical composition of phenyl isoxazolyl methylene-naphthalene-ether derivatives 甘莱制药有限公司 2021-06-04 CN disclosed
CN-112898289-A Compounds for modulating FXR activity and uses thereof 甘莱制药有限公司 2021-06-04 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230165843-A1 USE AND PHARMACEUTICAL COMPOSITION OF PHENYLISOXAZOLYL METHYLENE-NAPHTHALENE-ETHER DERIVATIVES VIM, CYP3A7, HAVCR2 NR1H4 116/4885HSD17B13 468/4885FABP1 39/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.