SCHEMBL25225632

SCHEMBL25225632

C[C@H](CC(=O)O)NS(=O)(=O)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
MMP1 P03956 1/20 0.55
MMP2 P08253 1/20 0.55
MMP9 P14780 1/20 0.55
MMP8 P22894 1/20 0.55
MMP13 P45452 1/20 0.55
THRB P10828 1/20 0.54
PKM P14618 1/20 0.50
HTT P42858 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.48
ALDH1A1 P00352 2/20 0.48
F2 P00734 1/20 0.48
PRSS1 P07477 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25272541 1.00 CA1 (0.55) CA1CA2MMP1MMP2MMP9
SCHEMBL30449084 0.87 CA1 (0.52) CA1CA2MMP1MMP2MMP9
SCHEMBL23779402 0.85 CA1 (0.59) CA1CA2MMP1MMP2MMP9
SCHEMBL14990813 0.85 CA1 (0.59) CA1CA2MMP1MMP2MMP9
SCHEMBL14990815 0.85 CA1 (0.59) CA1CA2MMP1MMP2MMP9
SCHEMBL5679181 0.85 CASP1 (0.64) CA1CA2MMP1MMP2MMP9
SCHEMBL25351582 0.84 CA1 (0.51) CA1CA2MMP1MMP2MMP9
SCHEMBL14094466 0.83 CA1 (0.56) CA1CA2MMP1MMP2MMP9
SCHEMBL12207830 0.82 CA1 (0.59) CA1CA2MMP1MMP2MMP9
SCHEMBL11527174 0.82 CA1 (0.59) CA1CA2MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024126617-A1 BIFUNCTIONAL COMPOUNDS FOR DEGRADING KINASES VIA UBIQUITIN PROTEOSOME PATHWAY CROSSFIRE ONCOLOGY HOLDING B.V. (NL) 2024-06-20 WO disclosed
WO-2023110970-A1 MACROCYCLIC BTK INHIBITORS NETHERLANDS TRANSLATIONAL RESEARCH CENTER HOLDING B.V (NL) 2023-06-22 WO disclosed
WO-2023110936-A1 REVERSIBLE MACROCYCLIC KINASE INHIBITORS NETHERLANDS TRANSLATIONAL RESEARCH CENTER HOLDING B.V (NL) 2023-06-22 WO disclosed