SCHEMBL25242491

SCHEMBL25242491

O=C1CCC(N2Cc3cc(CNC4CCN(Cc5ccccc5)CC4)ccc3C2=O)C(=O)N1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IKZF1 Q13422 6/20 0.63
IKZF2 Q9UKS7 10/20 0.61
CRBN Q96SW2 5/20 0.55
GSPT1 P15170 2/20 0.55
DDB1 Q16531 2/20 0.55
IKZF3 Q9UKT9 1/20 0.55
CYP2C19 P33261 1/20 0.54
KCNH2 Q12809 1/20 0.54
CSNK1A1 P48729 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25280863 0.95 IKZF1 (0.61) IKZF1IKZF2CRBNGSPT1DDB1
SCHEMBL25280864 0.95 IKZF1 (0.61) IKZF1IKZF2CRBNGSPT1DDB1
SCHEMBL25741173 0.90 IKZF2 (0.59) IKZF1IKZF2CRBNGSPT1DDB1
SCHEMBL25741174 0.90 IKZF2 (0.59) IKZF1IKZF2CRBNGSPT1DDB1
SCHEMBL61737 0.89 CRBN (0.62) IKZF1IKZF2CRBNGSPT1DDB1
SCHEMBL25741104 0.89 IKZF2 (0.59) IKZF1IKZF2CRBNGSPT1DDB1
SCHEMBL25235718 0.88 CRBN (0.58) IKZF1IKZF2CRBNGSPT1DDB1
SCHEMBL25741252 0.88 IKZF2 (0.57) IKZF1IKZF2CRBNGSPT1DDB1
SCHEMBL25741253 0.88 IKZF2 (0.57) IKZF1IKZF2CRBNGSPT1DDB1
SCHEMBL25742264 0.88 IKZF2 (0.57) IKZF1IKZF2CRBNGSPT1DDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4452414-A2 IKAROS ZINC FINGER FAMILY DEGRADERS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2024-10-30 EP disclosed
CN-118488946-A IKAROS zinc finger family degradation agent and application thereof 吉利德科学公司 2024-08-13 CN disclosed
US-20240124412-A1 IKAROS ZINC FINGER FAMILY DEGRADERS AND USES THEREOF GILEAD SCIENCES, INC. 2024-04-18 US disclosed
WO-2023122581-A2 IKAROS ZINC FINGER FAMILY DEGRADERS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2023-06-29 WO disclosed
WO-2023122581-A2 IKAROS ZINC FINGER FAMILY DEGRADERS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2023-06-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240124412-A1 IKAROS ZINC FINGER FAMILY DEGRADERS AND USES THEREOF IKZF2, IKZF1, IKZF3 IKZF1 2/4885IKZF2 1/4885CRBN 167/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.