SCHEMBL25244239

SCHEMBL25244239

CN(NC(=O)OC(C)(C)C)C(=O)c1cccc(F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
HTT P42858 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
OPRM1 P35372 1/20 0.41
OPRL1 P41146 1/20 0.41
PARP1 P09874 1/20 0.41
TSHR P16473 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25571223 0.85 ABCB1 (0.48) HDAC6PARP1MEN1KMT2ACYP3A4
SCHEMBL25571227 0.84 KMT2A (0.49) NPC1RAB9AHTTKDM4EALDH1A1
SCHEMBL25571225 0.83 RECQL (0.40) RAB9AHDAC6CTSSCTSKMEN1
SCHEMBL440962 0.83 AKT1 (0.49) NPC1RAB9AHTTTSHRCTSS
SCHEMBL25571224 0.83 ABCB1 (0.49) CES2CES1NPC1RAB9AHTT
SCHEMBL25571228 0.76 GAA (0.44) RAB9ALMNACYP3A4CYP2C9
SCHEMBL25571221 0.76 PPARG (0.41) CES2CES1NPC1RAB9AHDAC1
SCHEMBL25571226 0.75 LMNA (0.43) CTSSCTSKLMNA
SCHEMBL30437641 0.75 ESR1 (0.55) CES2CES1NPC1RAB9AHTT
SCHEMBL4224819 0.75 ESR1 (0.55) CES2CES1NPC1RAB9AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023097386-A1 SELECTIVE HDAC6-INHIBITING N-ACYLHYDRAZONE COMPOUNDS, METHODS FOR PRODUCING SAME, COMPOSITIONS, USES, TREATMENT METHODS AND KITS EUROFARMA LABORATÓRIOS S.A (BR) 2023-06-08 WO disclosed
WO-2023097386-A1 SELECTIVE HDAC6-INHIBITING N-ACYLHYDRAZONE COMPOUNDS, METHODS FOR PRODUCING SAME, COMPOSITIONS, USES, TREATMENT METHODS AND KITS EUROFARMA LABORATÓRIOS S.A (BR) 2023-06-08 WO disclosed