SCHEMBL2524460

SCHEMBL2524460

CC(NC(=O)O)n1ccc(-c2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 3/20 0.42
PHGDH O43175 6/20 0.42
ADORA1 P30542 2/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
MEN1 O00255 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
GRM5 P41594 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11623533 0.80 KMT2A (0.50) KMT2AKDM4EPHGDHADORA1CYP1A2
SCHEMBL17261556 0.78 ALDH1A1 (0.43) KMT2AKDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL17261466 0.78 ALDH1A1 (0.43) KMT2AKDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL17261471 0.78 ALDH1A1 (0.43) KMT2AKDM4EALDH1A1CYP1A2CYP2C9
SCHEMBL12777940 0.77 KMT2A (0.59) KMT2AKDM4EALDH1A1MEN1SMN1; SMN2
SCHEMBL17261487 0.76 MAPT (0.47) KMT2AKDM4EALDH1A1PHGDHADORA1
SCHEMBL17261473 0.75 AR (0.44) KMT2AKDM4ESMN1; SMN2
SCHEMBL17261490 0.75 AR (0.44) KMT2AKDM4ESMN1; SMN2
SCHEMBL11621690 0.75 KMT2A (0.45) KMT2AKDM4EALDH1A1PHGDHMEN1
SCHEMBL17261561 0.74 KMT2A (0.41) KMT2AKDM4EALDH1A1PHGDHADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2375899-A1 PIPERIDINE-CONTAINING COMPOUNDS AND USE THEREOF Array Biopharma, Inc. (US) 2011-10-19 EP disclosed
WO-2010080864-A1 PIPERIDINE-CONTAINING COMPOUNDS AND USE THEREOF ARRAY BIOPHARMA INC. (US) 2010-07-15 WO disclosed