SCHEMBL25257968

SCHEMBL25257968

C[Si](C)(C)CCOCn1cc(C(F)(F)F)c2nc(Cl)cnc21

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 9/20 0.46
PTPN1 P18031 1/20 0.34
P2RX7 Q99572 1/20 0.31
BRAF P15056 1/20 0.31
HDAC1 Q13547 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
HDAC5 Q9UQL6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25297250 0.86 DGAT1 (0.54) DGAT1PTPN1BRAF
SCHEMBL12372630 0.83 DGAT1 (0.38) DGAT1
SCHEMBL31512721 0.80 DGAT1 (0.45) DGAT1PTPN1P2RX7BRAF
SCHEMBL1352886 0.80 DGAT1 (0.38) DGAT1
SCHEMBL14738023 0.79 DGAT1 (0.42) DGAT1PTPN1
SCHEMBL25420967 0.79 DGAT1 (0.43) DGAT1PTPN1
SCHEMBL30461686 0.79 DGAT1 (0.43) DGAT1PTPN1
SCHEMBL20588479 0.78 DGAT1 (0.40) DGAT1PTPN1P2RX7
SCHEMBL25107078 0.77 DGAT1 (0.42) DGAT1PTPN1
SCHEMBL30205728 0.77 DGAT1 (0.42) DGAT1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118488947-A Condensed ring substituted six-membered heterocyclic compound, preparation method and application thereof 劲方医药科技(上海)有限公司 2024-08-13 CN disclosed
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed