SCHEMBL25286830

SCHEMBL25286830

CC(C)CC(NC(=O)C=Cc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 8/20 0.60
NOS3 P29474 7/20 0.60
NOS1 P29475 7/20 0.60
TAS1R3 Q7RTX0 2/20 0.60
TAS1R1 Q7RTX1 2/20 0.60
CASP1 P29466 1/20 0.53
CASP3 P42574 1/20 0.53
CASP7 P55210 1/20 0.53
CASP6 P55212 1/20 0.53
CASP8 Q14790 1/20 0.53
TDP1 Q9NUW8 2/20 0.51
MAPK1 P28482 4/20 0.49
ALDH1A1 P00352 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
MAPT P10636 6/20 0.48
KMT2A Q03164 3/20 0.48
ATM Q13315 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25286829 1.00 NOS2 (0.60) NOS2NOS3NOS1TAS1R3TAS1R1
SCHEMBL11902254 0.87 NOS2 (0.77) NOS2NOS3NOS1TAS1R3TAS1R1
SCHEMBL11902256 0.87 NOS2 (0.77) NOS2NOS3NOS1TAS1R3TAS1R1
SCHEMBL11902257 0.87 NOS2 (0.77) NOS2NOS3NOS1TAS1R3TAS1R1
SCHEMBL6015463 0.87 NOS2 (0.77) NOS2NOS3NOS1TAS1R3TAS1R1
SCHEMBL31389156 0.85 NOS2 (0.62) NOS2NOS3NOS1TAS1R3TAS1R1
SCHEMBL22994396 0.83 TDP1 (0.60) NOS2NOS3NOS1TAS1R3TAS1R1
SCHEMBL25286773 0.83 TDP1 (0.60) NOS2NOS3NOS1TAS1R3TAS1R1
SCHEMBL3947154 0.83 TDP1 (0.60) NOS2NOS3NOS1TAS1R3TAS1R1
SCHEMBL7313192 0.83 TDP1 (0.60) NOS2NOS3NOS1TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117751124-A Spiro oxindole compounds and application thereof in preparing antiviral protease inhibitor medicines 南京药石科技股份有限公司 2024-03-22 CN disclosed
WO-2023109926-A1 SPIROOXINDOLE COMPOUND AND USE THEREOF IN PREPARATION OF PROTEASE INHIBITOR AS ANTIVIRAL DRUG 南京药石科技股份有限公司 2023-06-22 WO disclosed