SCHEMBL25296196

SCHEMBL25296196

CC(C)(C)c1nn2c(I)ccc2cc1NC(=O)O

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.34
CDK8 P49336 1/20 0.33
MAPK14 Q16539 9/20 0.32
MAPK13 O15264 8/20 0.32
MAPK12 P53778 8/20 0.32
MAPK11 Q15759 8/20 0.32
JAK2 O60674 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
POLB P06746 1/20 0.31
PKM P14618 1/20 0.31
GAA P10253 1/20 0.30
ATM Q13315 1/20 0.30
SERPINE1 P05121 1/20 0.30
BRD9 Q9H8M2 1/20 0.30
DDR2 Q16832 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21543268 0.61 MEN1 (0.43) NPC1RAB9APOLBATM
SCHEMBL25302734 0.61 IGF1R (0.32) LMNACDK8MAPK14MAPK13MAPK12
SCHEMBL17836029 0.60 MEN1 (0.42) LMNANPC1RAB9APOLBGAA
SCHEMBL5847269 0.59 ENPP3 (0.33) NPC1RAB9APOLBGAA
SCHEMBL27228493 0.58 MAPT (0.34) LMNAPOLB
SCHEMBL28719439 0.58 NPC1 (0.47) LMNANPC1RAB9ASERPINE1
SCHEMBL18702740 0.58 NR1H4 (0.56) LMNANPC1RAB9ASERPINE1
SCHEMBL26607478 0.58 MAPT (0.50) LMNANPC1RAB9APKMGAA
SCHEMBL30218021 0.57 MAP3K5 (0.34) CDK8MAPK14MAPK13MAPK12MAPK11
SCHEMBL31160431 0.57 BACE1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250059196-A1 TRICYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF JIANGSU HANSOH PHARMACEUTICAL GROUP CO., LTD. (CN) 2025-02-20 US disclosed
EP-4458819-A1 TRICYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF Shanghai Hansoh Biomedical Co., Ltd. (CN) 2024-11-06 EP disclosed
WO-2023125877-A1 TRICYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海翰森生物医药科技有限公司 2023-07-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250059196-A1 TRICYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF WEE1, CYP51A1, WEE2 LMNA 2071/4885CDK8 171/4885MAPK14 1288/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.