SCHEMBL25304542

SCHEMBL25304542

N#Cc1cc(OCCC2CNCCO2)ccc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 8/20 0.40
SLC6A4 P31645 6/20 0.39
HTR2A P28223 4/20 0.39
SLC6A2 P23975 4/20 0.39
HTR2B P41595 2/20 0.39
SLC6A3 Q01959 2/20 0.39
ADRB2 P07550 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA2C P18825 1/20 0.39
HRH1 P35367 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
HTR3A P46098 1/20 0.37
KCNH2 Q12809 2/20 0.37
MKNK1 Q9BUB5 1/20 0.36
PRKACA P17612 1/20 0.36
PRKACG P22612 1/20 0.36
PRKACB P22694 1/20 0.36
EPHA2 P29317 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2761385 0.79 SLC6A4 (0.43) SLC6A4HTR2ASLC6A2HTR2BSLC6A3
SCHEMBL3657046 0.77 SLC6A2 (0.42) SLC6A4HTR2ASLC6A2HTR2BSLC6A3
SCHEMBL7216614 0.75 SLC6A4 (0.44) CHEK1SLC6A4HTR2ASLC6A2HTR2B
SCHEMBL5116224 0.74 SLC6A4 (0.43) CHEK1SLC6A4HTR2ASLC6A2HTR2B
SCHEMBL6941071 0.74 SLC6A4 (0.46) CHEK1SLC6A4HTR2ASLC6A2HTR2B
SCHEMBL4269340 0.72 TSHR (0.43) SLC6A4HTR2ASLC6A2HTR2BSLC6A3
SCHEMBL7349980 0.72 SLC6A4 (0.41) SLC6A4HTR2ASLC6A2HTR2BSLC6A3
SCHEMBL28467612 0.71 CHRNB2 (0.40) CHEK1SLC6A4HTR2ASLC6A2HTR2B
SCHEMBL7324975 0.71 HPGD (0.46) SLC6A4HTR2ASLC6A2HTR2BSLC6A3
SCHEMBL9385927 0.71 MEN1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134752-A1 DIARYL COMPOUND AS TUBULIN/SRC DUAL TARGET INHIBITOR 武汉人福创新药物研发中心有限公司 2023-07-20 WO disclosed