SCHEMBL25309201

SCHEMBL25309201

COCOc1cc(-c2ncc3c(N4CC5CCC(C4)N5C(=O)OC(C)(C)C)nc(OCC(OC)OC)nc3c2F)c2c(C#C[Si](C(C)C)(C(C)C)C(C)C)c(F)ccc2c1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KRAS P01116 20/20 0.39
MAPK3 P27361 1/20 0.37
MAPK1 P28482 1/20 0.37
RAF1 P04049 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25331029 0.93 KRAS (0.40) KRASMAPK3MAPK1RAF1
SCHEMBL30493773 0.93 KRAS (0.40) KRASMAPK3MAPK1RAF1
SCHEMBL31129488 0.93 KRAS (0.39) KRASMAPK3MAPK1RAF1
SCHEMBL31129339 0.92 KRAS (0.39) KRASMAPK3MAPK1RAF1
SCHEMBL31129721 0.92 KRAS (0.39) KRASMAPK3MAPK1RAF1
SCHEMBL31129533 0.92 KRAS (0.39) KRASMAPK3MAPK1RAF1
SCHEMBL30864045 0.92 KRAS (0.39) KRASMAPK3MAPK1RAF1
SCHEMBL31493993 0.92 KRAS (0.36) KRASMAPK3MAPK1RAF1
SCHEMBL31049086 0.91 KRAS (0.39) KRASMAPK3MAPK1RAF1
SCHEMBL25263547 0.91 KRAS (0.43) KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4655073-A2 CEREBLON-BASED KRAS DEGRADING PROTACS ANS USES RELATED THERETO Arvinas Operations, Inc. (US) 2025-12-03 EP disclosed
WO-2024159164-A2 CEREBLON-BASED KRAS DEGRADING PROTACS ANS USES RELATED THERETO ARVINAS OPERATIONS, INC. (US) 2024-08-02 WO disclosed
WO-2023141570-A9 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF KRAS ARVINAS OPERATIONS, INC. (US) 2024-06-27 WO disclosed
WO-2023141570-A2 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF KRAS ARVINAS OPERATIONS, INC. (US) 2023-07-27 WO disclosed