SCHEMBL25309474

SCHEMBL25309474

CC(C)(C)OC(=O)N1C2CCC1CN(c1ccc(C(F)(F)F)cn1)C2

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.57
HRH3 Q9Y5N1 3/20 0.51
KDM4E B2RXH2 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ABL1 P00519 1/20 0.50
LMNA P02545 1/20 0.50
HPGD P15428 1/20 0.50
HSD11B1 P28845 2/20 0.49
RET P07949 1/20 0.49
HCRTR1 O43613 3/20 0.48
HCRTR2 O43614 3/20 0.48
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
GPR119 Q8TDV5 1/20 0.47
MAPT P10636 3/20 0.47
ACACB O00763 2/20 0.46
SPR P35270 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30165102 1.00 HDAC1 (0.57) HDAC1HRH3KDM4ESMN1; SMN2ABL1
SCHEMBL18701834 0.86 KDM4E (0.54) HRH3KDM4ESMN1; SMN2ABL1LMNA
SCHEMBL24962970 0.85 GPR119 (0.57) HDAC1HSD11B1GPR119ACACB
SCHEMBL20468896 0.85 HDAC1 (0.60) HDAC1HRH3HSD11B1RETGPR119
SCHEMBL25310645 0.84 HDAC1 (0.57) HDAC1HSD11B1RETGPR119ACACB
SCHEMBL30510782 0.84 HDAC1 (0.57) HDAC1HSD11B1RETGPR119ACACB
SCHEMBL24428346 0.84 HDAC1 (0.59) HDAC1HSD11B1RETGPR119ACACB
SCHEMBL21262007 0.84 HDAC1 (0.59) HDAC1HSD11B1RETGPR119
SCHEMBL22909889 0.84 HDAC1 (0.59) HDAC1HSD11B1RETGPR119ACACB
SCHEMBL20456823 0.84 HDAC1 (0.62) HDAC1HSD11B1RETGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115745971-B PARP7 inhibitor and application thereof 北京华森英诺生物科技有限公司 2024-07-30 CN disclosed
WO-2023139536-A1 (4-PIPERAZIN-1YL)-4-ALKYL-PHTHALAZIN-1(2H)-ONE COMPOUNDS AS PARP7 INHIBITORS RHIZEN PHARMACEUTICALS AG (CH) 2023-07-27 WO disclosed