SCHEMBL25310064

SCHEMBL25310064

Cc1cc2ccc(Br)c(F)c2[nH]c1=O

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 16/20 0.42
ATAD2 Q6PL18 12/20 0.39
DAO P14920 2/20 0.38
DDO Q99489 2/20 0.38
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30482258 1.00 BRD4 (0.42) BRD4ATAD2DAODDOPARP1
SCHEMBL29266494 0.81 DAO (0.41) DAODDOPARP1
SCHEMBL30617953 0.81 DAO (0.41) DAODDOPARP1
SCHEMBL25604921 0.80 DAO (0.38) DAODDO
SCHEMBL30235048 0.80 DAO (0.38) DAODDO
SCHEMBL30617995 0.80 PARP1 (0.44) BRD4ATAD2DAODDOPARP1
SCHEMBL29266513 0.80 PARP1 (0.44) BRD4ATAD2DAODDOPARP1
SCHEMBL32673963 0.79 KDM4E (0.34)
SCHEMBL22199030 0.78 NQO2 (0.43) BRD4ATAD2
SCHEMBL25376520 0.76 BRD4 (0.41) BRD4ATAD2DAODDOPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260098024-A1 PARP1 INHIBITORS AND USES THEREOF XINTHERA INC (US) 2026-04-09 US disclosed
US-12384780-B2 PARP1 inhibitors and uses thereof XINTHERA, INC. (US) 2025-08-12 US disclosed
CN-120081844-A PARP1 inhibitors and uses thereof 新特拉有限公司 2025-06-03 CN disclosed
CN-118804916-B PARP1 inhibitors and uses thereof 新特拉有限公司 2025-04-01 CN disclosed
EP-4469449-A1 PARP1 INHIBITORS AND USES THEREOF Xinthera, Inc. (US) 2024-12-04 EP disclosed
EP-4466269-A1 PARP1 INHIBITORS AND USES THEREOF Xinthera, Inc. (US) 2024-11-27 EP disclosed
US-20240368162-A1 PARP1 INHIBITORS AND USES THEREOF XINTHERA, INC. 2024-11-07 US disclosed
CN-118804916-A PARP1 inhibitors and uses thereof 新特拉有限公司 2024-10-18 CN disclosed
CN-118510767-A PARP1 inhibitors and uses thereof 新特拉有限公司 2024-08-16 CN disclosed
US-11939329-B2 PARP1 inhibitors and uses thereof XINTHERA, INC. (US) 2024-03-26 US disclosed
WO-2024041643-A1 FUSED TRICYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF 江苏恒瑞医药股份有限公司 2024-02-29 WO disclosed
WO-2023146957-A1 PARP1 INHIBITORS AND USES THEREOF XINTHERA, INC. (US) 2023-08-03 WO disclosed
WO-2023146957-A1 PARP1 INHIBITORS AND USES THEREOF XINTHERA, INC. (US) 2023-08-03 WO disclosed
US-20230234952-A1 PARP1 INHIBITORS AND USES THEREOF XINTHERA, INC. 2023-07-27 US disclosed
US-20230234952-A1 PARP1 INHIBITORS AND USES THEREOF XINTHERA, INC. 2023-07-27 US disclosed
WO-2023141290-A1 PARP1 INHIBITORS AND USES THEREOF XINTHERA, INC. (US) 2023-07-27 WO disclosed
WO-2023141290-A1 PARP1 INHIBITORS AND USES THEREOF XINTHERA, INC. (US) 2023-07-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12384780-B2 PARP1 inhibitors and uses thereof PARP1, PARP11, PARP12 BRD4 37/4885ATAD2 1007/4885DAO 4505/4885
US-11939329-B2 PARP1 inhibitors and uses thereof PARP1, PARP11, PARP12 BRD4 37/4885ATAD2 1007/4885DAO 4505/4885
US-20230234952-A1 PARP1 INHIBITORS AND USES THEREOF PARP1, PARP11, PARP12 BRD4 37/4885ATAD2 1007/4885DAO 4505/4885
US-20260098024-A1 PARP1 INHIBITORS AND USES THEREOF PARP1, PARP11, PARP16 BRD4 28/4885ATAD2 1674/4885DAO 2762/4885
US-20240368162-A1 PARP1 INHIBITORS AND USES THEREOF PARP1, PARP11, PARP12 BRD4 37/4885ATAD2 1007/4885DAO 4505/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.