SCHEMBL22199030

SCHEMBL22199030

COc1ccc2cc(C)c(=O)[nH]c2c1F

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 5/20 0.43
CYP19A1 P11511 3/20 0.43
BRD4 O60885 10/20 0.41
ATAD2 Q6PL18 8/20 0.41
CNR2 P34972 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRIN2C Q14957 1/20 0.37
GRIN3A Q8TCU5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22198963 0.83 CYP19A1 (0.55) NQO2CYP19A1BRD4CNR2KDM4E
SCHEMBL22185224 0.82 ALDH1A1 (0.44) CNR2KDM4EALDH1A1
SCHEMBL22198968 0.81 NQO2 (0.43) NQO2CYP19A1BRD4ATAD2CNR2
SCHEMBL22184879 0.81 EIF4A3 (0.45) NQO2CYP19A1CNR2KDM4EALDH1A1
SCHEMBL25310064 0.78 BRD4 (0.42) BRD4ATAD2
SCHEMBL30482258 0.78 BRD4 (0.42) BRD4ATAD2
SCHEMBL5771632 0.76 GRIN2D (0.38) NQO2CYP19A1CNR2GRIN2DGRIN3B
SCHEMBL25262124 0.74 PARP1 (0.44) BRD4ATAD2KDM4EALDH1A1
SCHEMBL25310402 0.74 PARP1 (0.49) BRD4ATAD2KDM4EALDH1A1
SCHEMBL25376520 0.74 BRD4 (0.41) BRD4ATAD2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed