SCHEMBL25317145

SCHEMBL25317145

COC(=O)c1ccc(CN2CCN(Cc3ccc4c(c3)CN(C(=O)c3cc(C(C)C)c(OCc5ccccc5)cc3OCc3ccccc3)C4)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.52
HSP90AB1 P08238 2/20 0.52
HSP90B1 P14625 1/20 0.52
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
FAAH O00519 2/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PKM P14618 1/20 0.42
MAPK1 P28482 1/20 0.42
CHKA P35790 1/20 0.42
MAPT P10636 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31503222 1.00 HSP90AA1 (0.52) HSP90AA1HSP90AB1HSP90B1MEN1KMT2A
SCHEMBL25216919 0.93 HSP90AB1 (0.58) HSP90AA1HSP90AB1HSP90B1MEN1KMT2A
SCHEMBL25317220 0.93 HSP90AB1 (0.54) HSP90AA1HSP90AB1HSP90B1MEN1KMT2A
SCHEMBL384471 0.90 HSP90AB1 (0.64) HSP90AA1HSP90AB1HSP90B1MEN1KMT2A
SCHEMBL383809 0.89 HSP90AB1 (0.43) HSP90AA1HSP90AB1LMNAHDAC6
SCHEMBL31363033 0.89 HSP90AB1 (0.55) HSP90AA1HSP90AB1HSP90B1MEN1KMT2A
SCHEMBL25260723 0.87 HSP90AA1 (0.54) HSP90AA1HSP90AB1HSP90B1MEN1KMT2A
SCHEMBL16582202 0.87 HSP90AB1 (0.53) HSP90AA1HSP90AB1HSP90B1MEN1KMT2A
SCHEMBL30829338 0.87 HSP90AB1 (0.53) HSP90AA1HSP90AB1HSP90B1MEN1KMT2A
SCHEMBL31108361 0.87 HSP90AA1 (0.49) HSP90AA1HSP90AB1HSP90B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023140629-A1 2,7-SUBSTITUTED PYRROLO[2,1-F][1,2,4]TRIAZINE COMPOUND HAVING PROTEIN KINASE INHIBITORY ACTIVITY 닥터아이앤비(주) 2023-07-27 WO disclosed