SCHEMBL30829338

SCHEMBL30829338

CC(C)c1cc(C(=O)N2Cc3ccc(CN4CCNCC4)cc3C2)c(OCc2ccccc2)cc1OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 12/20 0.53
HSP90AA1 P07900 7/20 0.53
HSP90B1 P14625 1/20 0.53
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PARP1 P09874 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ABCB1 P08183 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16582202 1.00 HSP90AB1 (0.53) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A
Hydrochloric Acid SCHEMBL16569693 0.99 HSP90AB1 (0.52) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A
SCHEMBL25216919 0.93 HSP90AB1 (0.58) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A
SCHEMBL384471 0.91 HSP90AB1 (0.64) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A
SCHEMBL31363033 0.90 HSP90AB1 (0.55) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A
SCHEMBL25317220 0.89 HSP90AB1 (0.54) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A
SCHEMBL25260723 0.88 HSP90AA1 (0.54) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A
SCHEMBL31108384 0.88 HSP90AA1 (0.51) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A
SCHEMBL25271350 0.88 HSP90AA1 (0.51) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A
SCHEMBL25317145 0.87 HSP90AA1 (0.52) HSP90AB1HSP90AA1HSP90B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119100970-A Bivalent inhibitor based on heat shock protein 90 and preparation method and application thereof 中国药科大学 2024-12-10 CN claimed
CN-119100970-A Bivalent inhibitor based on heat shock protein 90 and preparation method and application thereof 中国药科大学 2024-12-10 CN disclosed
WO-2024034591-A1 HETEROCYCLIC COMPOUND FOR INHIBITING AND/OR INDUCING DEGRADATION OF KRAS PROTEIN アステラス製薬株式会社 2024-02-15 WO disclosed