SCHEMBL25329282

SCHEMBL25329282

CC(C)S(=O)(=O)c1ccccc1Nc1nc(NC2CCN(C(=O)OC(C)(C)C)C2)ncc1Cl

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 3/20 0.63
CDK7 P50613 2/20 0.63
PTK2 Q05397 6/20 0.56
ZAP70 P43403 1/20 0.55
ALK Q9UM73 9/20 0.54
MAPK3 P27361 1/20 0.53
ROS1 P08922 1/20 0.53
CDK2 P24941 2/20 0.53
CDK6 Q00534 2/20 0.53
AURKA O14965 1/20 0.53
NTRK1 P04629 1/20 0.53
IGF1R P08069 1/20 0.53
CDK4 P11802 1/20 0.53
EPHA1 P21709 1/20 0.53
CDK3 Q00526 1/20 0.53
CDK5 Q00535 1/20 0.53
CCNK O75909 1/20 0.53
CCNA2 P20248 1/20 0.53
CCND3 P30281 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25329276 1.00 CDK9 (0.63) CDK9CDK7PTK2ZAP70ALK
SCHEMBL29040469 0.95 CDK7 (0.62) CDK9CDK7PTK2ZAP70ALK
SCHEMBL23181216 0.95 CDK7 (0.62) CDK9CDK7PTK2ZAP70ALK
SCHEMBL30978800 0.95 CDK9 (0.68) CDK9CDK7PTK2ZAP70ALK
SCHEMBL29214366 0.95 CDK9 (0.68) CDK9CDK7PTK2ZAP70ALK
SCHEMBL25327813 0.91 PTK2 (0.56) CDK9CDK7PTK2ZAP70ALK
SCHEMBL25327808 0.91 PTK2 (0.56) CDK9CDK7PTK2ZAP70ALK
SCHEMBL25328917 0.90 PTK2 (0.57) CDK9CDK7PTK2ALKROS1
SCHEMBL25329554 0.90 PTK2 (0.57) CDK9CDK7PTK2ZAP70ALK
SCHEMBL25329544 0.90 PTK2 (0.57) CDK9CDK7PTK2ZAP70ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023143482-A1 2-AMINOPYRIMIDINE COMPOUND OR SALT, PREPARATION METHOD THEREFOR AND USE THEREOF 上海辉启生物医药科技有限公司 2023-08-03 WO disclosed