SCHEMBL25337040

SCHEMBL25337040

N#Cc1c(F)sc2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.44
ALDH1A1 P00352 7/20 0.42
KDM4E B2RXH2 4/20 0.42
MAPT P10636 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
GAA P10253 2/20 0.42
CACNA1B Q00975 1/20 0.42
APBA1 Q02410 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
HPGD P15428 1/20 0.33
IDO1 P14902 1/20 0.33
CASP1 P29466 2/20 0.33
ALOX15 P16050 2/20 0.33
MAPK1 P28482 2/20 0.33
POLB P06746 1/20 0.33
BRCA1 P38398 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31388718 0.78 GPR3 (0.46) GPR3ALDH1A1KDM4EMAPTMEN1
SCHEMBL4835675 0.76 GRM6 (0.46) GPR3ALDH1A1KDM4EMAPTMEN1
SCHEMBL29915175 0.76 GPR3 (0.44) GPR3ALDH1A1KDM4EMAPTMEN1
SCHEMBL23087421 0.76 GPR3 (0.44) GPR3ALDH1A1KDM4EMAPTMEN1
SCHEMBL12750484 0.76 GPR3 (0.44) GPR3ALDH1A1KDM4EMAPTMEN1
SCHEMBL1514430 0.76 GPR3 (0.44) GPR3ALDH1A1KDM4EMAPTMEN1
SCHEMBL14163676 0.76 GPR3 (0.40) GPR3ALDH1A1KDM4EMAPTMEN1
SCHEMBL32683687 0.74 CYP2A6 (0.35) MAPTGAAMAPK1POLBHTT
SCHEMBL23435972 0.72 GPR3 (0.40) GPR3ALDH1A1KDM4EMAPTMEN1
SCHEMBL29915197 0.72 GPR3 (0.40) GPR3ALDH1A1KDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260069605-A1 KRAS INHIBITORS INCYTE CORP (US) 2026-03-12 US disclosed
US-20260034126-A1 KRAS INHIBITORS INCYTE CORP (US) 2026-02-05 US disclosed
US-20260028357-A1 SUBSTITUTED HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC (US) 2026-01-29 US disclosed
US-12528828-B2 Substituted pyrido[4,3-d]pyrimidines as KRAS modulators ALTEROME THERAPEUTICS, INC. (US) 2026-01-20 US disclosed
US-20250346610-A1 SUBSTITUTED PYRIDO[4,3-d]PYRIMIDINES AS KRAS MODULATORS ALTEROME THERAPEUTICS INC (US) 2025-11-13 US disclosed
US-12466842-B2 Substituted pyrido [4,3-d]pyrimidines as KRAS modulators ALTEROME THERAPEUTICS, INC. (US) 2025-11-11 US disclosed
US-20250282799-A1 SUBSTITUTED PYRIDO[4,3-d]PYRIMIDINES AS KRAS MODULATORS ALTEROME THERAPEUTICS, INC. 2025-09-11 US disclosed
US-20250179093-A1 KRAS MODULATORS ALTEROME THERAPEUTICS, INC. 2025-06-05 US disclosed
CN-119119085-A Substituted pyrimido ring inhibitor and preparation method and application thereof 苏州泽璟生物制药股份有限公司 2024-12-13 CN disclosed
EP-4472980-A2 QUINAZOLINE PAN-KRAS INHIBITORS Mirati Therapeutics, Inc. (US) 2024-12-11 EP disclosed
WO-2023150284-A2 QUINAZOLINE PAN-KRAS INHIBITORS Mirati Therapeutics, Inc. (US) 2023-08-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250179093-A1 KRAS MODULATORS KRAS, NRAS, HRAS GPR3 2706/4885ALDH1A1 4071/4885KDM4E 3312/4885
US-20250346610-A1 SUBSTITUTED PYRIDO[4,3-d]PYRIMIDINES AS KRAS MODULATORS KRAS, NRAS, HRAS GPR3 1465/4885ALDH1A1 3593/4885KDM4E 1964/4885
US-12466842-B2 Substituted pyrido [4,3-d]pyrimidines as KRAS modulators KRAS, NRAS, HRAS GPR3 1465/4885ALDH1A1 3593/4885KDM4E 1964/4885
US-20260034126-A1 KRAS INHIBITORS KRAS, NRAS, HRAS GPR3 469/4885ALDH1A1 3023/4885KDM4E 4263/4885
US-20250282799-A1 SUBSTITUTED PYRIDO[4,3-d]PYRIMIDINES AS KRAS MODULATORS KRAS, NRAS, HRAS GPR3 1465/4885ALDH1A1 3593/4885KDM4E 1964/4885
US-12528828-B2 Substituted pyrido[4,3-d]pyrimidines as KRAS modulators KRAS, NRAS, HRAS GPR3 198/4885ALDH1A1 1854/4885KDM4E 4812/4885
US-20260069605-A1 KRAS INHIBITORS KRAS, NRAS, HRAS GPR3 442/4885ALDH1A1 966/4885KDM4E 4653/4885
US-20260028357-A1 SUBSTITUTED HETEROCYCLES AND USES THEREOF KRAS, HRAS, MYC GPR3 279/4885ALDH1A1 3875/4885KDM4E 4531/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.