SCHEMBL25345784

SCHEMBL25345784

Cc1cc2c(cc1O)CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.66
NR1H2 P55055 1/20 0.61
MAPK1 P28482 1/20 0.48
MAPT P10636 2/20 0.43
HDAC1 Q13547 1/20 0.41
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
MAP3K5 Q99683 2/20 0.40
ADORA1 P30542 2/20 0.40
IGF1R P08069 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
NAMPT P43490 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2122468 0.93 ESR2 (0.59) ESR2NR1H2MAPK1MAPTNPC1
SCHEMBL31054069 0.92 ESR2 (0.68) ESR2NR1H2MAPK1MAPTHDAC1
SCHEMBL5599903 0.92 ESR2 (0.72) ESR2NR1H2MAPK1MAPTHDAC1
SCHEMBL31359293 0.92 ESR2 (0.72) ESR2NR1H2MAPK1MAPTHDAC1
SCHEMBL18875035 0.85 NR1H2 (0.67) ESR2NR1H2MAPK1MAPTHDAC1
SCHEMBL21470912 0.85 ESR2 (0.64) ESR2NR1H2MAPK1MAPTHDAC1
SCHEMBL2805947 0.85 ESR2 (0.61) ESR2NR1H2MAPK1MAPTHDAC1
SCHEMBL23684548 0.85 ESR2 (0.68) ESR2NR1H2MAPK1MAPTHDAC1
SCHEMBL23684302 0.85 ESR2 (0.64) ESR2NR1H2MAPK1MAPTHDAC1
SCHEMBL4183582 0.85 NR1H2 (0.67) ESR2NR1H2MAPK1MAPTHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250179065-A1 HDAC6 INHIBITORS AND USES THEREOF EIKONIZO THERAPEUTICS, INC. (US) 2025-06-05 US disclosed
WO-2025101738-A1 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE PRELUDE THERAPEUTICS INCORPORATED (US) 2025-05-15 WO disclosed
US-20240174616-A1 HDAC6 INHIBITORS AND USES THEREOF EIKONIZO THERAPEUTICS, INC. (US) 2024-05-30 US disclosed
WO-2023150203-A1 HDAC6 INHIBITORS AND USES THEREOF EIKONIZO THERAPEUTICS, INC. (US) 2023-08-10 WO disclosed
WO-2023150203-A1 HDAC6 INHIBITORS AND USES THEREOF EIKONIZO THERAPEUTICS, INC. (US) 2023-08-10 WO disclosed
WO-2022169985-A1 HDAC6 INHIBITORS AND USES THEREOF EIKONIZO THERAPEUTICS, INC. (US) 2022-08-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240174616-A1 HDAC6 INHIBITORS AND USES THEREOF HDAC6, HDAC1, HDAC5 ESR2 3607/4885NR1H2 1754/4885MAPK1 2733/4885
US-20250179065-A1 HDAC6 INHIBITORS AND USES THEREOF HDAC6, HDAC1, HDAC5 ESR2 3607/4885NR1H2 1754/4885MAPK1 2733/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.