SCHEMBL2535397

SCHEMBL2535397

O=C(O)c1ccc(-c2cccc(F)c2)c(C(F)(F)F)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.57
AKR1C2 P52895 6/20 0.57
ADH5 P11766 1/20 0.49
PDE3B Q13370 2/20 0.46
PDE3A Q14432 2/20 0.46
SRD5A2 P31213 1/20 0.46
MRGPRX4 Q96LA9 1/20 0.45
ESR1 P03372 1/20 0.43
ESRRG P62508 1/20 0.43
AKR1C4 P17516 1/20 0.43
AKR1C1 Q04828 1/20 0.43
PLK4 O00444 1/20 0.43
AURKA O14965 1/20 0.43
DAPK3 O43293 1/20 0.43
CHEK2 O96017 1/20 0.43
CDK1 P06493 1/20 0.43
PIM1 P11309 1/20 0.43
CDK2 P24941 1/20 0.43
FLT4 P35916 1/20 0.43
KDR P35968 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL402398 0.86 ADH5 (0.58) AKR1C3AKR1C2ADH5SRD5A2EPHX2
SCHEMBL505879 0.81 AKR1C3 (0.56) AKR1C3AKR1C2ADH5PLK4AURKA
SCHEMBL23302210 0.81 ADH5 (0.63) AKR1C3AKR1C2ADH5SRD5A2EPHX2
SCHEMBL336261 0.81 ADH5 (0.54) AKR1C3AKR1C2ADH5SRD5A2P4HB
Hydrochloric Acid SCHEMBL28670680 0.80 ADH5 (0.61) AKR1C3AKR1C2ADH5SRD5A2EPHX2
Hydrochloric Acid SCHEMBL7740677 0.79 ADH5 (0.52) AKR1C3AKR1C2ADH5SRD5A2P4HB
Hydrochloric Acid SCHEMBL9229512 0.79 ADH5 (0.52) AKR1C3AKR1C2ADH5SRD5A2P4HB
SCHEMBL31268441 0.79 ADH5 (0.54) AKR1C3AKR1C2ADH5SRD5A2
SCHEMBL4539558 0.79 AKR1C3 (0.55) AKR1C3AKR1C2ADH5PDE3BPDE3A
SCHEMBL21271844 0.78 AKR1C3 (0.53) AKR1C3AKR1C2ADH5SRD5A2EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8273776-B2 Biphenyl oxadiazole derivatives as sphingosine-1-phosphate receptors modulators ALLERGAN, INC (US) 2012-09-25 US disclosed
US-20110257232-A1 BIPHENYL OXADIAZOLE DERIVATIVES AS SPHINGOSINE-1-PHOSPHATE RECEPTORS MODULATORS ALLERGAN, INC. (US) 2011-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110257232-A1 BIPHENYL OXADIAZOLE DERIVATIVES AS SPHINGOSINE-1-PHOSPHATE RECEPTORS MODULATORS S1PR3, S1PR1, S1PR2 AKR1C3 724/4885AKR1C2 1043/4885ADH5 2065/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.