SCHEMBL2536644

SCHEMBL2536644

COc1cc(-c2ccc3c(c2)C(C)(C)C(=O)N3)cc(OC)c1OC

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PGR P06401 13/20 0.63
MAP3K11 Q16584 2/20 0.60
PDE3B Q13370 5/20 0.51
PDE3A Q14432 5/20 0.51
PDE4A P27815 4/20 0.47
PDE4B Q07343 4/20 0.47
PDE4C Q08493 4/20 0.47
PDE4D Q08499 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2537789 0.77 MAP3K11 (0.66) PGRMAP3K11
SCHEMBL5225707 0.77 PGR (1.00) PGRPDE3BPDE3APDE4APDE4B
SCHEMBL719916 0.75 MAP3K11 (1.00) MAP3K11
SCHEMBL12886136 0.74 PGR (0.65) PGRPDE3BPDE3APDE4APDE4B
SCHEMBL10504098 0.74 MAP3K11 (0.47) PGRMAP3K11PDE3BPDE3APDE4A
SCHEMBL2270260 0.73 PGR (0.70) PGRPDE3BPDE3A
SCHEMBL12886131 0.73 PGR (0.63) PGRPDE3BPDE3APDE4APDE4B
SCHEMBL10373337 0.72 MAP3K11 (0.45) PGRMAP3K11
SCHEMBL10373335 0.72 PDE4A (0.58) MAP3K11PDE3BPDE3APDE4APDE4B
SCHEMBL3524585 0.71 PGR (0.85) PGRPDE3BPDE3APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379561-A2 MLK INHIBITORS AND METHODS OF USE University Of Rochester (US) 2011-10-26 EP disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed